SCHEMBL29183994

SCHEMBL29183994

COC(=O)CCCCN1CCN(c2nc(-c3ccc(N)cc3)nc(N3CCOCC3)n2)CC1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 18/20 0.58
MTOR P42345 17/20 0.58
PIK3R1 P27986 1/20 0.58
PIK3CG P48736 15/20 0.50
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
DRD2 P14416 1/20 0.45
DRD3 P35462 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29183799 0.89 PIK3CA (0.61) PIK3CAMTORPIK3R1PIK3CGHDAC3
SCHEMBL29183819 0.88 PIK3CA (0.60) PIK3CAMTORPIK3R1PIK3CGHDAC3
SCHEMBL29183975 0.88 PIK3CA (0.58) PIK3CAMTORPIK3R1PIK3CGHDAC3
SCHEMBL29183979 0.87 HDAC1 (0.60) PIK3CAMTORPIK3R1PIK3CGHDAC3
SCHEMBL29183992 0.87 PIK3CA (0.57) PIK3CAMTORPIK3R1PIK3CGHDAC3
SCHEMBL29183995 0.86 DRD2 (0.43) PIK3CAMTORPIK3R1PIK3CGHDAC3
SCHEMBL29183797 0.81 MTOR (0.65) PIK3CAMTORPIK3R1PIK3CG
SCHEMBL29184046 0.78 PIK3CA (0.64) PIK3CAMTORPIK3R1PIK3CG
SCHEMBL28714705 0.78 DRD4 (0.49) DRD2
SCHEMBL29183796 0.77 PIK3CA (0.63) PIK3CAMTORPIK3R1PIK3CGHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117777042-A Triazine hydroxamic acid derivative and preparation method and application thereof 长沙医学院 2024-03-29 CN disclosed