SCHEMBL29200480

SCHEMBL29200480

CCc1cccc(Nc2ccnc3cc(C(F)(F)F)ccc23)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 3/20 0.57
APP P05067 1/20 0.54
NR4A2 P43354 1/20 0.54
GSK3A P49840 3/20 0.48
GSK3B P49841 3/20 0.48
CLK4 Q9HAZ1 2/20 0.48
ACVR1 Q04771 1/20 0.48
MST1R Q04912 1/20 0.48
TYRO3 Q06418 1/20 0.48
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
EPHB6 O15197 1/20 0.47
RIPK2 O43353 1/20 0.47
ABL1 P00519 1/20 0.47
LCK P06239 1/20 0.47
EPHA1 P21709 1/20 0.47
EPHA8 P29322 1/20 0.47
TXK P42681 1/20 0.47
COQ8A Q8NI60 1/20 0.47
NLK Q9UBE8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29200458 0.82 GAK (0.64) GAKGSK3AGSK3BCLK4EPHB6
SCHEMBL28845692 0.82 FADS1 (0.66) GAKAPPNR4A2GSK3AGSK3B
SCHEMBL28845712 0.82 EGFR (0.66) GAKGSK3AGSK3BCLK4EPHB6
SCHEMBL28845637 0.80 DNMT1 (0.52) GAKGSK3AGSK3BCLK4ACVR1
SCHEMBL29200469 0.80 GAK (0.55) GAKGSK3AGSK3BCLK4ACVR1
SCHEMBL11553078 0.79 KDM4E (0.50) GAKAPPMAPKAPK2
SCHEMBL28845634 0.79 GAK (0.55) GAKGSK3AGSK3BCLK4ACVR1
SCHEMBL28845679 0.79 GAK (0.50) GAKAPPNR4A2GSK3AGSK3B
SCHEMBL29089850 0.78 GAK (0.65) GAKGSK3AGSK3BCLK4EPHB6
SCHEMBL11557265 0.78 MAPKAPK2 (0.47) GAKMAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN claimed