SCHEMBL29201425

SCHEMBL29201425

Cc1c(-c2ccccc2)ccc(F)c1CBr

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
DHODH Q02127 2/20 0.38
PTGER2 P43116 1/20 0.38
KAT6A Q92794 1/20 0.36
ERBB2 P04626 1/20 0.35
ESR2 Q92731 1/20 0.34
PTGS1 P23219 4/20 0.34
MEN1 O00255 2/20 0.34
PTGS2 P35354 2/20 0.34
KMT2A Q03164 2/20 0.34
FABP2 P12104 1/20 0.34
TSHR P16473 1/20 0.34
AKR1C4 P17516 1/20 0.34
ADRA2B P18089 1/20 0.34
CHRM3 P20309 1/20 0.34
HTR2C P28335 1/20 0.34
DRD3 P35462 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28433870 0.84 PDCD1 (0.50) PDCD1CD274DHODHPTGER2KAT6A
SCHEMBL10990692 0.81 ALOX5AP (0.37) PTGER2PTGS1MEN1PTGS2KMT2A
SCHEMBL10972725 0.81 PDCD1 (0.43) PDCD1CD274ERBB2ESR2PTGS1
SCHEMBL16554648 0.80 PDCD1 (0.42) PDCD1CD274ERBB2ESR2PTGS1
SCHEMBL4486456 0.75 PDCD1 (0.42) PDCD1CD274DHODHKAT6AESR2
SCHEMBL5501718 0.74 ALDH1A1 (0.44) ESR2TSHRHPGDCYP2A6ALDH1A1
SCHEMBL15856379 0.73 PDCD1 (0.41) PDCD1CD274KAT6AESR2PTGS1
SCHEMBL27456057 0.72 POLB (0.40) PDCD1CD274KAT6AESR2PTGS1
SCHEMBL10985670 0.71 GRIN1 (0.40) PDCD1CD274KAT6AESR2PTGS1
SCHEMBL9792869 0.71 PDCD1 (0.54) PDCD1CD274ESR2PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117729921-A Compounds and methods as PD1/PD-L1 inhibitors 朱比兰特普罗德尔有限公司 2024-03-19 CN disclosed