SCHEMBL16554648

SCHEMBL16554648

Cc1c(-c2ccccc2)ccc(I)c1CBr

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.42
CD274 Q9NZQ7 1/20 0.42
ERBB2 P04626 1/20 0.36
ESR2 Q92731 1/20 0.35
PARP10 Q53GL7 1/20 0.35
PARP11 Q9NR21 1/20 0.35
ALDH1A1 P00352 3/20 0.33
CYP2A6 P11509 1/20 0.33
CYP2B6 P20813 1/20 0.33
MAPK1 P28482 1/20 0.33
PTGS1 P23219 1/20 0.33
TRPA1 O75762 1/20 0.32
TSHR P16473 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
AKT1 P31749 1/20 0.32
AKT2 P31751 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
SQOR Q9Y6N5 1/20 0.31
KDM4E B2RXH2 2/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10972725 0.83 PDCD1 (0.43) PDCD1CD274ERBB2ESR2PARP10
SCHEMBL29201425 0.80 PDCD1 (0.41) PDCD1CD274ERBB2ESR2PARP10
SCHEMBL5501718 0.75 ALDH1A1 (0.44) ESR2ALDH1A1CYP2A6MAPK1TRPA1
SCHEMBL9792869 0.72 PDCD1 (0.54) PDCD1CD274ESR2PARP10PARP11
Ammonia Solution, Strong SCHEMBL9346396 0.72 CD274 (0.47) PDCD1CD274ERBB2ESR2PARP10
SCHEMBL6067573 0.72 PDCD1 (0.39) PDCD1CD274ESR2PARP10PARP11
SCHEMBL14963930 0.70 PTGS1 (0.39) PDCD1CD274ERBB2ESR2ALDH1A1
SCHEMBL20500632 0.70 SQOR (0.38) PDCD1CD274ALDH1A1TSHRSQOR
SCHEMBL24051152 0.70 PDCD1 (0.53) PDCD1CD274ESR2PARP10PARP11
SCHEMBL24570750 0.70 ESR2 (0.45) PDCD1CD274ESR2PARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041822-A1 COMPOUNDS USEFUL AS IMMUNOMODULATORS Bristol-Myers Squibb Company (US) 2016-07-13 EP disclosed
WO-2015034820-A1 COMPOUNDS USEFUL AS IMMUNOMODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2015-03-12 WO disclosed