SCHEMBL29207709

SCHEMBL29207709

COC1CCN(c2ncc(-c3ccc(OCc4ccccc4)nc3OCc3ccccc3)cn2)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.42
OGA O60502 1/20 0.41
CYP11B2 P19099 1/20 0.40
EHMT2 Q96KQ7 2/20 0.39
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAOB P27338 1/20 0.38
AOC3 Q16853 1/20 0.37
PDE10A Q9Y233 1/20 0.37
GRM5 P41594 2/20 0.37
KIT P10721 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30801285 0.86 ALDH1A1 (0.49) HRH4CYP11B2ALDH1A1SMN1; SMN2AOC3
SCHEMBL24671246 0.86 PDE10A (0.40) HRH4CYP11B2ALDH1A1SMN1; SMN2PDE10A
SCHEMBL30066309 0.86 PDE10A (0.40) HRH4CYP11B2ALDH1A1SMN1; SMN2PDE10A
SCHEMBL25200347 0.81 GPR119 (0.40) HRH4AOC3GRM5
SCHEMBL31306744 0.76 PDE10A (0.40) HRH4ALDH1A1SMN1; SMN2PDE10A
SCHEMBL29872807 0.75 PRMT5 (0.41) PDE10A
SCHEMBL23459570 0.75 PRMT5 (0.41) PDE10A
SCHEMBL31692696 0.75 NT5E (0.40) HRH4GRM5
SCHEMBL23984155 0.74 PRMT5 (0.38) HRH4CYP11B2ALDH1A1SMN1; SMN2GRM5
SCHEMBL25504062 0.74 CNR2 (0.44) HRH4CYP11B2ALDH1A1SMN1; SMN2PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117693502-A Compounds for inhibiting or degrading ITK, compositions comprising the same, methods of making the same, and methods of using the same 纽力克斯治疗公司 2024-03-12 CN disclosed