SCHEMBL29213784

SCHEMBL29213784

COC(=O)c1ccc([C@]2(Cc3ccccc3)CC(=C3CC3)CCN2C(=O)O)cc1F

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.34
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
TACR1 P25103 1/20 0.32
TACR3 P29371 1/20 0.32
PLA2G2A P14555 1/20 0.32
ALDH1A1 P00352 4/20 0.32
KDM4E B2RXH2 3/20 0.32
GAA P10253 3/20 0.32
LMNA P02545 1/20 0.32
ATM Q13315 1/20 0.31
ALOX15 P16050 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29213867 0.90 HTR6 (0.34) HTR6CHRNB4CHRNA3MEN1KMT2A
SCHEMBL29213845 0.70 CA1 (0.38) MEN1KMT2AALDH1A1KDM4E
SCHEMBL3742265 0.66 KMT2A (0.36) MEN1KMT2AALDH1A1LMNAATM
SCHEMBL29213766 0.65 PARP1 (0.42) ALDH1A1
SCHEMBL18030873 0.65 PLA2G2A (0.53) HTR6PLA2G2AALDH1A1KDM4EGAA
SCHEMBL31474027 0.63 CA12 (0.40) KMT2AALDH1A1KDM4EGAALMNA
SCHEMBL16709817 0.63 SMN1; SMN2 (0.50) MEN1KMT2AALDH1A1KDM4EGAA
SCHEMBL23163640 0.62 ALDH1A1 (0.41) KMT2AALDH1A1KDM4EGAAATM
SCHEMBL176858 0.62 MAOB (0.59) ALDH1A1LMNA
SCHEMBL1484340 0.61 KMT2A (0.54) MEN1KMT2AALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118043314-A Benzazepine heteroaromatic ring derivative and application thereof in medicine 西藏海思科制药有限公司 2024-05-14 CN disclosed
WO-2023020566-A1 BENZO NITROGEN-CONTAINING HETEROAROMATIC RING DERIVATIVE AND USE THEREOF IN MEDICINE 四川海思科制药有限公司 2023-02-23 WO disclosed