SCHEMBL29228294

SCHEMBL29228294

CC1(C)CCc2cc(-c3ccccc3OC(F)(F)F)ccc2C1OC(N)=O

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 18/20 0.45
SCN10A Q9Y5Y9 1/20 0.43
CYP2C9 P11712 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
OPRD1 P41143 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29228194 0.92 SCN9A (0.43) SCN9ASCN10ACYP2C9CYP3A4CYP2D6
SCHEMBL28828402 0.90 SCN9A (0.44) SCN9ASCN10ACYP2C9CYP3A4CYP2D6
SCHEMBL29228270 0.87 SCN9A (0.40) SCN9ASCN10AOPRD1
SCHEMBL29228173 0.85 PARP1 (0.38) OPRD1
SCHEMBL29228243 0.85 DHODH (0.42)
SCHEMBL29228295 0.85 PPIB (0.41) SCN9A
SCHEMBL29228364 0.83 DHODH (0.39) SCN9AOPRD1
SCHEMBL29228256 0.83 EGFR (0.38) SCN9A
SCHEMBL29228205 0.83 ABCB1 (0.39)
SCHEMBL29228212 0.82 PGR (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114746422-B Derivatives having 1,2,3, 4-tetrahydronaphthalene moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-03-12 CN claimed
CN-114746422-A Novel derivatives having 1,2,3, 4-tetrahydronaphthalene moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2022-07-12 CN claimed
CN-114746422-B Derivatives having 1,2,3, 4-tetrahydronaphthalene moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-03-12 CN disclosed
CN-114746422-A Novel derivatives having 1,2,3, 4-tetrahydronaphthalene moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2022-07-12 CN disclosed