SCHEMBL29228596

SCHEMBL29228596

COc1ccc(I)c(C(=O)OC(C)(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 2/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
CYP3A4 P08684 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
ELANE P08246 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31707789 0.87 NPC1 (0.45) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL23963498 0.83 ELANE (0.50) ELANE
SCHEMBL28430334 0.83 KDM4E (0.60) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13387623 0.81 HPGD (0.48) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL21395373 0.81 NOS2 (0.48) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL4405887 0.81 CPS1 (0.44) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL271075 0.80 GABRA1 (0.44) KDM4EMAPTALDH1A1ABCG2HPGD
SCHEMBL2982404 0.80 CISD2 (0.40) CYP2C9CYP2C19NPSR1GABRA1GABRG2
SCHEMBL23963502 0.80 ELANE (0.40) KDM4EMAPTMAPK1ELANEPOLB
SCHEMBL4688965 0.79 KDM4E (0.45) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118027018-A Tetrahydrocyclopentyl [ c ] pyrrole methyl ketone derivative, preparation method and application thereof 江苏恩华药业股份有限公司 2024-05-14 CN disclosed