SCHEMBL29244161

SCHEMBL29244161

FC(F)(F)Oc1ccc(C2=N[CH]CS2)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.43
SCN5A Q14524 7/20 0.39
KCNH2 Q12809 3/20 0.38
SCN1A P35498 3/20 0.38
SCN2A Q99250 3/20 0.38
SCN9A Q15858 2/20 0.38
SCN8A Q9UQD0 2/20 0.38
SCN10A Q9Y5Y9 2/20 0.38
PIM1 P11309 2/20 0.38
PIM2 Q9P1W9 1/20 0.38
NOTUM Q6P988 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
PIP4K2A P48426 1/20 0.38
PTGS2 P35354 2/20 0.37
PTGS1 P23219 1/20 0.37
KIF11 P52732 1/20 0.36
GALR1 P47211 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29244152 0.81 DYRK1A (0.43) KCNH2SCN10APIM1PIM2GALR1
SCHEMBL29244205 0.71 SCN9A (0.40) SCN9A
SCHEMBL2040458 0.69
SCHEMBL254957 0.68 MAPT (0.56) NISCHPIM1PIM2NOTUMKIF11
SCHEMBL10224674 0.67 NISCH (0.38) NISCHSCN5AKCNH2SCN1ASCN2A
SCHEMBL16878883 0.66 NISCH (0.49) NISCHSCN5ASCN1ASCN2APIM2
SCHEMBL8111753 0.65 KIF11 (0.56) NISCHSCN5ASCN1ASCN2AKIF11
SCHEMBL14893848 0.65 NISCH (0.44) NISCHPIM1PIM2NOTUMPTGS2
SCHEMBL28616564 0.64 KMT2A (0.53) SCN5ASCN1ASCN2ANOTUM
SCHEMBL306823 0.64 KIF11 (0.50) NISCHSCN5ASCN1ASCN2AKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118290434-A Spiropiperidine derivative containing alpha-methylene-gamma-butyrolactone, preparation method and application thereof 南开大学 2024-07-05 CN claimed
CN-118290434-A Spiropiperidine derivative containing alpha-methylene-gamma-butyrolactone, preparation method and application thereof 南开大学 2024-07-05 CN disclosed