SCHEMBL292480

SCHEMBL292480

[CH2]C1=CCc2ccccc2O1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.48
MAOB P27338 2/20 0.48
GAA P10253 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
OXTR P30559 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL292788 0.76 MAOA (0.50) MAOAMAOBGAANPSR1NPC1
SCHEMBL30356272 0.76 MAOA (0.50) MAOAMAOBGAANPSR1NPC1
SCHEMBL11391339 0.74 MAOA (0.48) MAOAMAOBGAANPSR1NPC1
SCHEMBL1862899 0.74 MAOA (0.48) MAOAMAOBGAANPSR1NPC1
SCHEMBL57273 0.74 MAOA (0.48) MAOAMAOBGAANPSR1NPC1
SCHEMBL753891 0.74 MAOA (0.48) MAOAMAOBGAANPSR1NPC1
SCHEMBL2006248 0.74 MAOA (0.48) MAOAMAOBGAANPSR1NPC1
SCHEMBL1939933 0.74 MAOA (0.48) MAOAMAOBGAANPSR1NPC1
SCHEMBL758245 0.74 MAOA (0.48) MAOAMAOBGAANPSR1NPC1
SCHEMBL30140866 0.74 MAOA (0.48) MAOAMAOBGAANPSR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6617281-B1 Substituted acylamino phenyl uracils BAYER AKTIENGESELLSCHAFT (DE) 2003-09-09 US claimed
EP-1095028-A1 SUBSTITUTED ACYLAMINO PHENYL URACILS BAYER AG (DE) 2001-05-02 EP claimed
WO-2000002867-A1 SUBSTITUTED ACYLAMINO PHENYL URACILS BAYER AKTIENGESELLSCHAFT (DE) 2000-01-20 WO claimed
EP-3131897-B1 FACTOR IXA INHIBITORS MERCK SHARP & DOHME (US) 2022-06-15 EP disclosed
EP-3131896-B1 FACTOR IXA INHIBITORS MERCK SHARP & DOHME (US) 2019-01-30 EP disclosed
US-9969724-B2 Factor IXa inhibitors MERCK SHARP & DOHME CORP. (US) 2018-05-15 US disclosed
US-9808445-B2 Factor IXa inhibitors MERCK SHARP & DOHME CORP. (US) 2017-11-07 US disclosed
US-20170129880-A1 FACTOR IXa INHIBITORS MERCK SHARP & DOHME LLC 2017-05-11 US disclosed
EP-3131896-A1 FACTOR IXA INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-02-22 EP disclosed
EP-3131897-A1 FACTOR IXA INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-02-22 EP disclosed
US-20170027916-A1 FACTOR IXa INHIBITORS MERCK SHARP & DOHME CORP. (US) 2017-02-02 US disclosed
EP-1555267-A1 2,3-DIHYDRO-6-NITROIMIDAZO 2,1-b OXAZOLES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-07-20 EP disclosed
CN-1193020-C Process for preparing amic acid esters IHARA CHEMICAL IND CO (JP) 2005-03-16 CN disclosed
US-6617281-B1 Substituted acylamino phenyl uracils BAYER AKTIENGESELLSCHAFT (DE) 2003-09-09 US disclosed
US-6576765-B2 Process for preparing amic acid esters IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2003-06-10 US disclosed
US-20030032667-A1 PROCESS FOR PREPARING AMIC ACID ESTERS IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2003-02-13 US disclosed
CN-1366523-A Process for preparing amic acid esters IHARA CHEMICAL IND CO (JP) 2002-08-28 CN disclosed
EP-1182199-A1 PROCESS FOR PREPARING AMIC ACID ESTERS IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2002-02-27 EP disclosed
EP-1095028-A1 SUBSTITUTED ACYLAMINO PHENYL URACILS BAYER AG (DE) 2001-05-02 EP disclosed
WO-2000002867-A1 SUBSTITUTED ACYLAMINO PHENYL URACILS BAYER AKTIENGESELLSCHAFT (DE) 2000-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170129880-A1 FACTOR IXa INHIBITORS F9, F12, TFPI MAOA 116/4885MAOB 250/4885GAA 210/4885
US-20170027916-A1 FACTOR IXa INHIBITORS F9, F12, TFPI MAOA 116/4885MAOB 250/4885GAA 210/4885
US-20030032667-A1 PROCESS FOR PREPARING AMIC ACID ESTERS MCCC2, EMC1, GANC MAOA 656/4885MAOB 779/4885GAA 853/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.