SCHEMBL2925835

SCHEMBL2925835

Cc1cnc(Cl)nc1-c1cc2cccc(-c3ccncc3)c2s1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.37
GSK3B P49841 3/20 0.35
CDK2 P24941 1/20 0.35
CDC7 O00311 3/20 0.35
DBF4 Q9UBU7 3/20 0.35
MAPK14 Q16539 2/20 0.35
MAPK11 Q15759 1/20 0.35
CYP17A1 P05093 2/20 0.33
CYP1A2 P05177 2/20 0.33
MAPK9 P45984 1/20 0.33
MAPK10 P53779 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
TDO2 P48775 1/20 0.32
WNT1 P04628 1/20 0.32
TGFBR1 P36897 1/20 0.32
PDK1 Q15118 2/20 0.31
PDK2 Q15119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2923179 0.87 TDO2 (0.39) PDE10AGSK3BCDK2CDC7DBF4
SCHEMBL2922754 0.81 ADORA1 (0.39) PDE10AGSK3BCDK2CDC7DBF4
SCHEMBL2927723 0.81 CA12 (0.30) CA12CA1CA2CA9PDK1
SCHEMBL2870401 0.79 BTK (0.33) CA12CA1CA2CA9PDK1
SCHEMBL29809458 0.78 PDE10A (0.48) PDE10AGSK3BCDK2CDC7DBF4
SCHEMBL594142 0.75 CA12 (0.30) CA12CA1CA2CA9PDK1
SCHEMBL2919757 0.74 BTK (0.32) FGFR1
SCHEMBL13829027 0.73 MAPK14 (0.40) MAPK14MAPK11PDK1PDK2PDK3
SCHEMBL3963838 0.73 PIK3CD (0.41) CA1CA2CA9
SCHEMBL394127 0.72 LIMK1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101563342-B Imidazolidinonyl aminopyrimidine compounds for the treatment' of cancer LILLY CO ELI 2012-09-05 CN disclosed
EP-2125793-B1 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2010-09-01 EP disclosed
CN-101563342-A Imidazolidinonyl aminopyrimidine compounds for the treatment' of cancer LILLY CO ELI (US) 2009-10-21 CN disclosed