SCHEMBL292734

SCHEMBL292734

COc1ccc(F)cc1C(C)(C)CC(O)(Cc1cc2cc(C(=O)N3CCC(O)C3)ccc2[nH]1)C(F)(F)F

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 20/20 0.67
NR3C2 P08235 16/20 0.67
PGR P06401 14/20 0.67
CYP3A4 P08684 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4555748 0.99 NR3C1 (0.65) NR3C1NR3C2PGRCYP3A4
SCHEMBL292319 0.95 NR3C1 (0.69) NR3C1NR3C2PGRCYP3A4
SCHEMBL4558038 0.92 NR3C1 (0.63) NR3C1NR3C2PGRCYP3A4
SCHEMBL293515 0.89 NR3C1 (0.73) NR3C1NR3C2PGRCYP3A4
SCHEMBL292292 0.89 NR3C1 (0.72) NR3C1NR3C2PGRCYP3A4
SCHEMBL292075 0.88 NR3C1 (0.71) NR3C1NR3C2PGRCYP3A4
SCHEMBL291658 0.87 NR3C1 (0.70) NR3C1NR3C2PGRCYP3A4
SCHEMBL292257 0.87 NR3C1 (0.70) NR3C1NR3C2PGRCYP3A4
SCHEMBL14158607 0.84 NR3C1 (0.65) NR3C1NR3C2PGRCYP3A4
SCHEMBL290758 0.83 NR3C1 (0.82) NR3C1NR3C2PGRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050176706-A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-08-11 US claimed
US-8741897-B2 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2014-06-03 US disclosed
US-8741897-B2 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2014-06-03 US disclosed
US-8741897-B2 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2014-06-03 US disclosed
EP-2056799-B1 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING GLAUCOMA OR PROGRESSION THEREOF BAUSCH & LOMB (US) 2013-07-31 EP disclosed
EP-2203160-B1 PHARMACOLOGICAL ADJUNCTIVE TREATMENT ASSOCIATED WITH GLAUCOMA FILTRATION SURGERY BAUSCH & LOMB (US) 2013-07-17 EP disclosed
EP-2190431-B1 COMPOSITIONS COMPRISING A DISSOCIATED GLUCOCORTICOID RECEPTOR AGONIST FOR TREATING OR CONTROLLING ANTERIOR-SEGMENT INFLAMMATION BAUSCH & LOMB (US) 2013-07-03 EP disclosed
EP-2364707-B1 Compositions and methods for treating, controlling, reducing, or ameliorating infections and sequelae thereof BAUSCH & LOMB (US) 2013-04-03 EP disclosed
US-20120316199-A1 COMPOSITIONS AND METHODS FOR TREATING, CONTROLLING, REDUCING, OR AMELIORATING INFLAMMATORY PAIN SOLTA MEDICAL IRELAND LIMITED (IE) 2012-12-13 US disclosed
US-20120065228-A1 COMPOSITIONS AND METHODS FOR TREATING, CONTROLLING, REDUCING, OR AMELIORATING OCULAR INFLAMMATORY WITH LOWER RISK OF INCREASED INTRAOCULAR PRESSURE SOLTA MEDICAL, INC. 2012-03-15 US disclosed
WO-2005030213-A1 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-04-07 WO disclosed
CN-1158063-C Rinse-off water-in-oil-in-water compositions ˹��������ͼ˹�����µ� 2004-07-21 CN disclosed
US-20030161796-A1 Composition for treating hair UNILEVER HOME & PERSONAL CARE USA, DIVISION OF CONOPCO, INC. 2003-08-28 US disclosed
US-6022547-A EXTERNAL AQUEOUS PHASE AND INTERNAL PHASE COMPRISING A PRIMARY WATER-IN-OIL EMULSION, WHEREIN THE PRIMARY EMULSION COMPRISES A FIRST TOPICALLY-ACTIVE COMPOUND, A SURFACTANT PHASE, OIL PHASE AND WATER HELENE CURTIS, INC. (US) 2000-02-08 US disclosed
US-5942216-A COMPRISING AN EXTERNAL AQUEOUS PHASE OF A SURFACTANT CAPABLE OF FORMIG LIQUID CRYSTALS AS AN EMULSIFIER; THE INTERNAL WATER-IN OIL EMULSION HAVING A TOPICALLY-ACTIVE COMPOUND AND SURFACTANT AND OIL PHASES; HAIR AND SKIN TREATMENTS HELENE CURTIS, INC. (US) 1999-08-24 US disclosed
US-5656280-A CONTAINING A SURFACTANT BLEND FOR STABILITY AND A TOPICALLY-ACTIVE COMPOUND HELENE CURTIS, INC. (US) 1997-08-12 US disclosed
CN-1138982-A Rinse-off water-in-oil-in-water compositions CURTIS HELENE IND INC (US) 1997-01-01 CN disclosed
US-5589177-A OIL SOLUBLE SILICONES WITH WATER FOR EMULSIONS FOR TOPICAL APPLICATION AND HAIR FIXATIVES HELENE CURTIS, INC. (US) 1996-12-31 US disclosed
EP-0717978-A2 Rinse-off water-in-oil-in-water compositions HELENE CURTIS INC. (US) 1996-06-26 EP disclosed
EP-0715842-A2 Water-in-oil-in-water compositions HELENE CURTIS INC. (US) 1996-06-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176706-A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof NR3C1, NR3C2, MC2R NR3C1 1/4885NR3C2 2/4885PGR 95/4885
US-20120065228-A1 COMPOSITIONS AND METHODS FOR TREATING, CONTROLLING, REDUCING, OR AMELIORATING OCULAR INFLAMMATORY WITH LOWER RISK OF INCREASED INTRAOCULAR PRESSURE PTGIR, NR3C1, PTGDR NR3C1 2/4885NR3C2 11/4885PGR 272/4885
US-20120316199-A1 COMPOSITIONS AND METHODS FOR TREATING, CONTROLLING, REDUCING, OR AMELIORATING INFLAMMATORY PAIN PTGIR, MC2R, NR3C1 NR3C1 3/4885NR3C2 18/4885PGR 220/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.