Diketopiperazine

Diketopiperazine

SCHEMBL29279043

O=C1CNC(=O)CN1.c1ccc2c(c1)CCC2

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.53
TSHR P16473 1/20 0.52
CYP2A6 P11509 2/20 0.48
MAOB P27338 2/20 0.48
MAOA P21397 1/20 0.48
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
NPC1 O15118 1/20 0.42
MAPK13 O15264 1/20 0.42
MAPK12 P53778 1/20 0.42
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
PNMT P11086 1/20 0.41
CD44 P16070 1/20 0.41
HTR2C P28335 1/20 0.41
PDPK1 O15530 1/20 0.41
PARP1 P09874 1/20 0.41
PARP10 Q53GL7 1/20 0.41
PARP11 Q9NR21 1/20 0.41
AHR P35869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydantoin SCHEMBL7756713 0.84 MAPT (0.52) MAPTTSHRCYP2A6MAOBMAOA
Hydantoin SCHEMBL5442026 0.79 TSHR (0.50) MAPTTSHRCYP2A6MAOBMAOA
SCHEMBL8119999 0.77 MAPT (0.70) MAPTTSHRCYP2A6MAOBMAOA
SCHEMBL2062062 0.77 NPC1 (0.52) MAPTTSHRCYP2A6MAOBCA12
SCHEMBL3057782 0.77 TSHR (0.86) MAPTTSHRCYP2A6MAOBMAOA
SCHEMBL29354295 0.77
SCHEMBL9662 0.77
SCHEMBL451157 0.77 TSHR (0.86) MAPTTSHRCYP2A6MAOBMAOA
SCHEMBL23766313 0.77 MAPT (0.67) MAPTTSHRCYP2A6MAOBMAOA
SCHEMBL5193435 0.76 ALOX15 (0.57) MAPTCA12CA9NPC1MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110914240-B Norbornenone compounds releasing carbon monoxide 奥塔哥创新有限公司 2024-02-20 CN disclosed
CN-110914240-A Norbornene ketone compounds releasing carbon monoxide 奥塔哥创新有限公司 2020-03-24 CN disclosed