SCHEMBL29280405

SCHEMBL29280405

C#Cc1ccc(N2CC(C(N)=O)C2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.48
RORC P51449 1/20 0.39
NOTUM Q6P988 4/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
MGLL Q99685 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
WDR91 A4D1P6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2297674 0.78 NOTUM (0.58) RORCNOTUMKDM4EALDH1A1LMNA
SCHEMBL5053496 0.75 CHKA (0.44) RORCNOTUMMEN1KMT2A
SCHEMBL6132253 0.70 MAPT (0.51) AKR1C3KDM4EALDH1A1MAPTHRH3
SCHEMBL6132255 0.70 MAPT (0.51) AKR1C3KDM4EALDH1A1MAPTHRH3
SCHEMBL15532039 0.70 PARP1 (0.46) RORCNOTUMJAK3
SCHEMBL30188574 0.69 SMN1; SMN2 (0.37) RORCNOTUMKDM4EALDH1A1POLB
SCHEMBL30932001 0.68 CTSK (0.43) AKR1C3KMT2AJAK3
SCHEMBL14662156 0.68 AKR1C3 (0.50) AKR1C3RORCNOTUMKDM4EMAPT
SCHEMBL2636602 0.68 NOTUM (0.54) RORCNOTUMALDH1A1MAPTWDR91
SCHEMBL15531010 0.68 NOTUM (0.36) RORCNOTUMKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117751113-A Aromatic acetylene derivative and preparation method and application thereof 浙江海正药业股份有限公司 2024-03-22 CN disclosed
WO-2023011573-A1 AROMATIC ACETYLENE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江海正药业股份有限公司 2023-02-09 WO disclosed