SCHEMBL29285015

SCHEMBL29285015

O=C(O)c1ccc(CNC(=O)c2ccccc2I)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.64
NR1H4 Q96RI1 6/20 0.61
EPHX2 P34913 4/20 0.61
KMT2A Q03164 3/20 0.59
SMN1; SMN2 Q16637 1/20 0.57
CYP1A2 P05177 1/20 0.56
CYP2C19 P33261 1/20 0.56
ALDH1A1 P00352 2/20 0.54
HPGD P15428 2/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
POLB P06746 1/20 0.54
HSD17B10 Q99714 1/20 0.54
CTDSP1 Q9GZU7 1/20 0.54
MAPT P10636 1/20 0.53
LMNA P02545 1/20 0.53
GAA P10253 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
METAP2 P50579 1/20 0.51
CHRNB2 P17787 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11319016 0.89 KMT2A (0.69) APEX1KMT2ACYP1A2CYP2C19HPGD
SCHEMBL12700348 0.86 APEX1 (0.87) APEX1NR1H4EPHX2KMT2ASMN1; SMN2
SCHEMBL28053361 0.83 APEX1 (0.57) APEX1KMT2ASMN1; SMN2CYP1A2CYP2C19
SCHEMBL28053295 0.83 KMT2A (0.70) APEX1KMT2ASMN1; SMN2CYP1A2CYP2C19
SCHEMBL4182426 0.83 ALDH1A1 (0.62) APEX1KMT2ASMN1; SMN2CYP1A2CYP2C19
SCHEMBL28053365 0.83 HPGD (0.68) APEX1KMT2ASMN1; SMN2ALDH1A1HPGD
SCHEMBL16088749 0.82 APEX1 (0.69) APEX1NR1H4EPHX2KMT2ASMN1; SMN2
SCHEMBL1060622 0.82 HPGD (0.71) APEX1NR1H4EPHX2KMT2ASMN1; SMN2
SCHEMBL8226871 0.82 APEX1 (0.64) APEX1NR1H4EPHX2KMT2ASMN1; SMN2
SCHEMBL27752218 0.82 KMT2A (0.64) APEX1NR1H4EPHX2KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118255731-A Synthesis method of biguanide derivative 湖北玖天生物医药科技有限公司 2024-06-28 CN claimed
CN-118255731-A Synthesis method of biguanide derivative 湖北玖天生物医药科技有限公司 2024-06-28 CN disclosed