SCHEMBL29289652

SCHEMBL29289652

NCc1ccc2c(c1)C(=O)N=C2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
ROCK1 Q13464 1/20 0.35
PDPK1 O15530 1/20 0.35
ST14 Q9Y5Y6 1/20 0.34
CSNK2A1 P68400 3/20 0.33
LOXL2 Q9Y4K0 3/20 0.32
LOX P28300 1/20 0.32
LOXL3 P58215 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29289892 0.85 GAA (0.41) GAAPKMCA12CA1CA2
SCHEMBL31098567 0.85 GAA (0.41) GAAPKMCA12CA1CA2
SCHEMBL29024953 0.81 CA12 (0.35) CA12CA1CA2CA3CA4
SCHEMBL21715527 0.72 TDP2 (0.43)
SCHEMBL30740450 0.69 AR (0.39) PDPK1
SCHEMBL21573719 0.67 NPC1 (0.55) GAAPKMCA12CA1CA2
SCHEMBL15889108 0.67 PPOX (0.50) GAAPKMPDPK1
SCHEMBL21715511 0.67 ALDH1A1 (0.36)
SCHEMBL30740688 0.67 TDP2 (0.46) GAACA12CA1CA2CA4
SCHEMBL20300390 0.67 CHEK1 (0.38) CA12CA1CA2CA3CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113563245-B Substituted pyrrolidines and their use in medicine 广东东阳光药业股份有限公司 2024-10-15 CN disclosed
CN-113563245-A Substituted pyrrolidine compounds and application thereof in medicines 广东东阳光药业有限公司 2021-10-29 CN disclosed