SCHEMBL2929059

SCHEMBL2929059

CCc1nc(NC(=O)O)sc1SC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 3/20 0.51
TMIGD3 P0DMS9 1/20 0.48
ADORA1 P30542 1/20 0.48
ALDH1A1 P00352 6/20 0.39
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.36
RAB9A P51151 2/20 0.36
HTT P42858 2/20 0.36
HSD17B10 Q99714 2/20 0.36
GPER1 Q99527 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
HPGD P15428 1/20 0.36
KAT8 Q9H7Z6 1/20 0.36
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9570975 0.70 ALDH1A1 (0.50) ADORA1ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL11222481 0.68 MAPT (0.45) FBP1ALDH1A1MEN1KMT2ARAB9A
SCHEMBL773032 0.66 LCK (0.61)
SCHEMBL2175442 0.66 SMN1; SMN2 (0.34) FBP1ALDH1A1LMNASMN1; SMN2RAB9A
SCHEMBL16238270 0.66 RAB9A (0.64) ALDH1A1NPSR1RXFP1MEN1KMT2A
SCHEMBL11225698 0.66 MAPT (0.43) FBP1ALDH1A1MEN1KMT2ARAB9A
SCHEMBL1743735 0.66 ALDH1A1 (0.39) ALDH1A1NPSR1RXFP1MEN1KMT2A
SCHEMBL16742808 0.65 ALDH1A1 (0.34) ALDH1A1MEN1KMT2ASMN1; SMN2RAB9A
SCHEMBL7144220 0.65 MEN1 (0.40) ALDH1A1LMNANPSR1RXFP1MEN1
SCHEMBL11224332 0.65 MAPT (0.40) FBP1ALDH1A1RXFP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227468-A1 AMINOTHIAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-09-15 EP disclosed
WO-2009068467-A1 AMINOTHIAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-06-04 WO disclosed