SCHEMBL2929658

SCHEMBL2929658

Cc1ccc(C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)c(-c2ccc(F)c(C)c2)c1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 11/20 0.36
HCRTR1 O43613 7/20 0.36
GRIN2B Q13224 1/20 0.34
CYP3A4 P08684 2/20 0.33
KDM1A O60341 2/20 0.33
MAPK14 Q16539 1/20 0.33
SRC P12931 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2926254 0.92 HCRTR2 (0.40) HCRTR2HCRTR1KDM1A
SCHEMBL2931971 0.90 HCRTR1 (0.36) HCRTR2HCRTR1
SCHEMBL2924236 0.89 KDM1A (0.35) HCRTR2HCRTR1KDM1A
SCHEMBL2929505 0.86 HCRTR2 (0.43) HCRTR2HCRTR1
SCHEMBL2925064 0.86 HCRTR2 (0.43) HCRTR2HCRTR1
SCHEMBL2924875 0.86 HCRTR2 (0.37) HCRTR2HCRTR1HTR2A
SCHEMBL2929656 0.85 HCRTR2 (0.37) HCRTR2HCRTR1GRIN2BCYP3A4
SCHEMBL2926155 0.85 HDAC7 (0.43) HCRTR2HCRTR1
SCHEMBL2930272 0.84 CHRM1 (0.46) HCRTR2HCRTR1
SCHEMBL2928985 0.84 GRM2 (0.35) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP claimed
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed