SCHEMBL2929754

SCHEMBL2929754

FC(F)(F)c1ccc(C2C[N]CC(c3ncc(-c4ccccc4)s3)C2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.40
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
SLC6A3 Q01959 3/20 0.38
KIF11 P52732 1/20 0.36
KDM1A O60341 3/20 0.35
MAOB P27338 3/20 0.35
PSEN1 P49768 2/20 0.35
PSEN2 P49810 2/20 0.35
APH1B Q8WW43 2/20 0.35
NCSTN Q92542 2/20 0.35
APH1A Q96BI3 2/20 0.35
PSENEN Q9NZ42 2/20 0.35
SCN2A Q99250 2/20 0.34
MET P08581 1/20 0.34
HTR2C P28335 2/20 0.33
HDAC4 P56524 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KDM4E B2RXH2 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3963514 0.81 TRPV1 (0.41) TRPV1SLC6A2SLC6A4SLC6A3PSEN1
SCHEMBL641993 0.75 F2R (0.61) TRPV1KIF11
SCHEMBL29786817 0.70 KDR (0.46) TRPV1SLC6A2SLC6A4SLC6A3
SCHEMBL4677035 0.69 KDR (0.41) TRPV1SLC6A2SLC6A4SLC6A3
SCHEMBL26255820 0.68 KDR (0.44) TRPV1SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL26976668 0.66 KDR (0.41) SLC6A2SLC6A4SLC6A3
SCHEMBL4875916 0.65 SLC6A2 (0.58) SLC6A2SLC6A4SLC6A3
SCHEMBL4677044 0.65 CHRNB2 (0.53) SLC6A2SLC6A4SLC6A3
SCHEMBL3723293 0.65 HTR2C (0.50) SLC6A3KIF11KDM1AMAOBHTR2C
SCHEMBL1765207 0.64 MLYCD (0.46) TRPV1SLC6A2SLC6A4SLC6A3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227466-A2 HETEROARYL-SUBSTITUTED PIPERIDINES Bayer Schering Pharma Aktiengesellschaft (DE) 2010-09-15 EP disclosed
WO-2009068214-A2 HETEROARYL-SUBSTITUTED PIPERIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-06-04 WO disclosed