SCHEMBL2930255

SCHEMBL2930255

C=Cc1ccc(CN2CCC(N(C)C)CC2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 1/20 0.45
PRKCD Q05655 1/20 0.45
PARP1 P09874 4/20 0.42
PARP2 Q9UGN5 1/20 0.40
TNKS O95271 1/20 0.39
KMT2A Q03164 1/20 0.39
MAP4K4 O95819 1/20 0.39
FLT3 P36888 1/20 0.38
MERTK Q12866 1/20 0.38
GAS6 Q14393 1/20 0.38
KCNH2 Q12809 2/20 0.38
GPR119 Q8TDV5 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
DRD2 P14416 2/20 0.37
HTR2A P28223 2/20 0.37
SIGMAR1 Q99720 2/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
LTA4H P09960 1/20 0.37
DRD1 P21728 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18291574 0.82 PARP1 (0.44) PRKCQPRKCDPARP1PARP2TNKS
SCHEMBL20255406 0.81 DRD2 (0.45) PRKCQPRKCDPARP1PARP2TNKS
SCHEMBL29475483 0.81 TRPV6 (0.51) PARP1PARP2TNKSKMT2AMAP4K4
SCHEMBL18291711 0.81 MAP4K4 (0.44) PRKCQPRKCDPARP1PARP2TNKS
SCHEMBL2933977 0.81 TRPV6 (0.51) PARP1PARP2TNKSKMT2AMAP4K4
SCHEMBL30786240 0.79 HRH3 (0.52) HRH3
SCHEMBL2929383 0.79 LMNA (0.50) KMT2AHRH3
SCHEMBL20249124 0.78 KCNH2 (0.47) PARP1PARP2TNKSKMT2AMAP4K4
SCHEMBL20037688 0.78 PARP1 (0.42) PARP1PARP2TNKSKMT2AMAP4K4
SCHEMBL17646031 0.76 HRH3 (0.53) HRH3LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP disclosed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO disclosed