Cgs-19281A

Cgs-19281A

SCHEMBL2930783

COc1ccc2c3c([nH]c2c1)C=NCC3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.58
CYP3A4 P08684 4/20 0.58
CYP2D6 P10635 4/20 0.58
ALDH1A1 P00352 4/20 0.58
HTR2C P28335 4/20 0.58
HTR7 P34969 4/20 0.58
MEN1 O00255 3/20 0.58
CASP1 P29466 3/20 0.58
KMT2A Q03164 3/20 0.58
HPGD P15428 3/20 0.58
HSD17B10 Q99714 3/20 0.58
HTR6 P50406 3/20 0.58
GLA P06280 2/20 0.58
TSHR P16473 2/20 0.58
CASP7 P55210 2/20 0.58
POLB P06746 2/20 0.58
GAA P10253 2/20 0.58
MAPT P10636 2/20 0.58
HTR2A P28223 2/20 0.58
RECQL P46063 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cgs-19281A SCHEMBL29769895 1.00 KDM4E (0.58) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C
SCHEMBL30921653 0.89 KDM4E (0.58) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C
SCHEMBL28631444 0.89 KDM4E (0.58) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C
Harmaline SCHEMBL9481244 0.88 KDM4E (0.80) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C
SCHEMBL1655707 0.81 KDM4E (0.52) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C
SCHEMBL678673 0.73 HTR2C (0.54) KDM4EALDH1A1HTR2CHTR7MEN1
Harmaline SCHEMBL29626541 0.73 KDM4E (1.00) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C
Harmaline SCHEMBL199260 0.73 KDM4E (1.00) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C
SCHEMBL1520427 0.72 KDM4E (0.74) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C
Harmaline SCHEMBL1360259 0.72 KDM4E (0.97) KDM4ECYP3A4CYP2D6ALDH1A1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107141288-B Evodiamine compounds and preparation method and application thereof 中山大学 2019-12-27 CN disclosed
EP-2227233-A2 IDO INHIBITORS Newlink Genetics (US) 2010-09-15 EP disclosed
WO-2009073620-A2 IDO INHIBITORS NEWLINK GENETICS (US) 2009-06-11 WO disclosed