SCHEMBL29311604

SCHEMBL29311604

CN(C)CCOc1cc(N)c(NO)cc1Br

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.45
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
HRH3 Q9Y5N1 5/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
ROCK2 O75116 1/20 0.38
UTS2R Q9UKP6 2/20 0.37
LMNA P02545 1/20 0.35
ESR1 P03372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29311606 0.84 HTR7 (0.44) HTR7CYP1A2CYP2D6CYP2C19HRH3
SCHEMBL25319735 0.83 HTR7 (0.54) HTR7CYP1A2CYP2D6CYP2C19HRH3
SCHEMBL31078181 0.72 KDM4E (0.49) HTR7CYP1A2CYP2D6CYP2C19HRH3
SCHEMBL25321839 0.72 KDM4E (0.49) HTR7CYP1A2CYP2D6CYP2C19HRH3
SCHEMBL7399293 0.71 HTR7 (0.60) HTR7CYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL30058042 0.69 HTR7 (0.53) HTR7CYP1A2CYP2D6CYP2C19HRH3
SCHEMBL23875588 0.69 HTR7 (0.53) HTR7CYP1A2CYP2D6CYP2C19HRH3
SCHEMBL1986857 0.69 HTR7 (0.49) HTR7CYP1A2CYP2D6CYP2C19HRH3
SCHEMBL25794425 0.69 HTR7 (0.49) HTR7CYP1A2CYP2D6CYP2C19HRH3
SCHEMBL1974546 0.69 KDM4E (0.44) HTR7CYP1A2CYP2D6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024141443-A1 BENZIMIDAZOLE DERIVATIVES USEFUL AS SIK MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2024-07-04 WO disclosed