SCHEMBL29311685

SCHEMBL29311685

Clc1ccc(OC2CCN(C3COC3)CC2)nn1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 1/20 0.37
HRH3 Q9Y5N1 9/20 0.35
KCNH2 Q12809 1/20 0.35
LRRK2 Q5S007 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
PDCD1LG2 Q9BQ51 1/20 0.33
CD274 Q9NZQ7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30986469 1.00 MAP3K12 (0.37) MAP3K12HRH3KCNH2LRRK2ABCG2
SCHEMBL29311693 0.83 MAP3K12 (0.39) MAP3K12HRH3KCNH2
SCHEMBL25318985 0.80 CHRNB2 (0.37) KCNH2
SCHEMBL30508902 0.80 CHRNB2 (0.37) KCNH2
SCHEMBL31110184 0.78 CHRNB2 (0.40)
SCHEMBL30986545 0.78 HRH3 (0.42) HRH3KCNH2LRRK2
SCHEMBL17654119 0.75 LMNA (0.55)
SCHEMBL16292286 0.74 HRH3 (0.44) MAP3K12HRH3KCNH2
SCHEMBL16292314 0.74 HRH3 (0.44) MAP3K12HRH3KCNH2
SCHEMBL12949577 0.74 LOX (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024141443-A1 BENZIMIDAZOLE DERIVATIVES USEFUL AS SIK MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2024-07-04 WO disclosed