SCHEMBL29314042

SCHEMBL29314042

CNc1ncc(C#N)c(NCC(C)(C)CO)n1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.45
AURKA O14965 1/20 0.39
CHEK1 O14757 1/20 0.38
LRRK2 Q5S007 9/20 0.38
CDK1 P06493 1/20 0.38
KDR P35968 1/20 0.38
SYK P43405 1/20 0.37
PRKCQ Q04759 5/20 0.35
PRKCD Q05655 5/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29313462 0.86 LRRK2 (0.39) AURKACHEK1LRRK2SYKPRKCQ
SCHEMBL29313773 0.81 CCNA2 (0.46) AURKALRRK2CDK1KDRSYK
SCHEMBL18293973 0.79 PRKCQ (0.56) CHEK1PRKCQPRKCD
SCHEMBL16842117 0.77 PRKCQ (0.63) PRKCQPRKCD
SCHEMBL29313606 0.73 PTK2 (0.40) AURKALRRK2SYKPRKCQ
SCHEMBL23019347 0.73 PRKCQ (0.41) AURKALRRK2SYKPRKCQ
SCHEMBL29315063 0.73 LRRK2 (0.35) AURKALRRK2CDK1KDRSYK
SCHEMBL4770519 0.71 AURKA (0.46) AURKACHEK1LRRK2CDK1KDR
SCHEMBL29313552 0.71 PTK2 (0.43) AURKALRRK2SYKPRKCQPRKCD
SCHEMBL29314061 0.70 PDE4A (0.39) AURKALRRK2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed