SCHEMBL29313606

SCHEMBL29313606

CNc1ncc(C#N)c(NCc2ncccn2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.40
PTK2B Q14289 1/20 0.40
CLK1 P49759 1/20 0.39
CLK2 P49760 1/20 0.39
CLK3 P49761 1/20 0.39
DYRK1A Q13627 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
SYK P43405 1/20 0.39
AURKA O14965 1/20 0.38
SIRT5 Q9NXA8 1/20 0.38
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
PRKCQ Q04759 6/20 0.37
EGFR P00533 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
LRRK2 Q5S007 3/20 0.36
PGK1 P00558 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29313537 0.84 PTK2 (0.56) PTK2PTK2BSYKKDM4EGAA
SCHEMBL29313552 0.81 PTK2 (0.43) PTK2PTK2BSYKAURKAPRKCQ
SCHEMBL29313542 0.81 ALDH1A1 (0.54) CLK4SIRT5KDM4EPGK1
SCHEMBL29313615 0.80 VNN1 (0.47) PTK2PTK2BSYKAURKASIRT5
SCHEMBL29315097 0.79 MAP3K8 (0.43) PTK2PTK2BSYKAURKASIRT5
SCHEMBL29313621 0.78 PTK2 (0.41) PTK2PTK2BSYKAURKASIRT5
SCHEMBL29315070 0.78 MAP3K8 (0.45) PTK2PTK2BCLK2CLK4SYK
SCHEMBL29313773 0.77 CCNA2 (0.46) SYKAURKASIRT5KDM4EPRKCQ
SCHEMBL29315063 0.75 LRRK2 (0.35) SYKAURKASIRT5PRKCQLRRK2
SCHEMBL29314042 0.73 NUDT1 (0.45) SYKAURKAPRKCQLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed