SCHEMBL29314047

SCHEMBL29314047

CN(C(=O)Oc1c(C(F)(F)F)cc(C(F)(F)F)c(Cl)c1-c1cnco1)c1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 7/20 0.36
POLQ O75417 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
IMPDH2 P12268 2/20 0.34
IMPDH1 P20839 1/20 0.34
AAK1 Q2M2I8 1/20 0.33
GPR119 Q8TDV5 3/20 0.32
P2RX7 Q99572 1/20 0.32
SCD O00767 1/20 0.31
SCD5 Q86SK9 1/20 0.31
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29314040 0.90 POLQ (0.36) LIPEPOLQMEN1KMT2AIMPDH2
SCHEMBL29314049 0.87 POLQ (0.34) LIPEPOLQMEN1KMT2AIMPDH2
SCHEMBL29314044 0.82 POLQ (0.42) LIPEPOLQIMPDH2IMPDH1AAK1
SCHEMBL30847644 0.73 POLQ (0.41) LIPEPOLQMEN1KMT2AKDM4E
SCHEMBL29314063 0.70 POLQ (0.39) LIPEPOLQIMPDH2IMPDH1GPBAR1
SCHEMBL29314384 0.69 POLQ (0.52) LIPEPOLQKDM4ENPC1ALDH1A1
SCHEMBL29314067 0.68 POLQ (0.43) LIPEPOLQ
SCHEMBL30847596 0.68 POLQ (0.50) LIPEPOLQMEN1KMT2AMAPK1
SCHEMBL29314388 0.68 POLQ (0.50) LIPEPOLQMEN1KMT2AALDH1A1
SCHEMBL31009186 0.67 POLQ (0.44) LIPEPOLQGPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed