SCHEMBL29314783

SCHEMBL29314783

CNc1ncc(C#N)c(-c2ccnc(OC)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.47
CDK1 P06493 6/20 0.47
LRRK2 Q5S007 2/20 0.45
KDM5A P29375 1/20 0.45
ACVR2A P27037 4/20 0.41
TGFBR1 P36897 4/20 0.41
TGFBR2 P37173 4/20 0.41
AAK1 Q2M2I8 2/20 0.41
ADORA1 P30542 3/20 0.41
ADORA2A P29274 2/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA2B P29275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16116775 0.82 ADORA1 (0.56) KDRCDK1LRRK2KDM5AACVR2A
SCHEMBL29314691 0.74 ADORA1 (0.63) KDRCDK1ADORA1ADORA2AADORA2B
SCHEMBL29314862 0.74 ADORA1 (0.64) KDRCDK1ADORA1ADORA2AADORA2B
SCHEMBL29315373 0.73 KDR (0.48) KDRCDK1ADORA1ADORA2A
SCHEMBL29314680 0.72 KDR (0.45) KDRCDK1ADORA1ADORA2AADORA2B
SCHEMBL25597187 0.70 IDH1 (0.45) KDRCDK1LRRK2
SCHEMBL29314732 0.69 KDR (0.61) KDRCDK1ADORA1ADORA2A
SCHEMBL23019360 0.69 KDR (0.41) KDRCDK1ADORA1ADORA2A
SCHEMBL20446788 0.69 AAK1 (0.55) LRRK2KDM5AACVR2ATGFBR2AAK1
SCHEMBL29314718 0.68 CYP11B1 (0.48) KDRCDK1ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed