SCHEMBL29315915

SCHEMBL29315915

CC(C)(C)OC(=O)n1cc(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2CC(=O)O)cn1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.37
AGBL2 Q5U5Z8 1/20 0.36
SCD O00767 1/20 0.36
SCN9A Q15858 2/20 0.34
CACNA1B Q00975 2/20 0.34
CACNA1C Q13936 2/20 0.34
CACNA1H O95180 1/20 0.34
TACR1 P25103 2/20 0.34
CACNA1G O43497 1/20 0.34
GCGR P47871 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
RXRA P19793 5/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
STS P08842 1/20 0.32
POLQ O75417 1/20 0.32
RXRB P28702 4/20 0.32
RXRG P48443 4/20 0.32
GPR17 Q13304 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31009206 0.90 ROCK2 (0.36) ROCK2SCDSCN9ACACNA1BCACNA1C
SCHEMBL29316280 0.84 ROCK2 (0.39) ROCK2SCDSCN9ACACNA1BCACNA1C
SCHEMBL31009207 0.81 POLQ (0.50) ROCK2SCDSCN9APOLQ
SCHEMBL22353102 0.73 ROCK2 (0.42) ROCK2SCDTACR1STS
SCHEMBL16895188 0.73 ROCK2 (0.45) ROCK2SCDSCN9ANR1H2STS
SCHEMBL29315913 0.72 ROCK1 (0.39) ROCK2AGBL2GCGRPTGDR2RXRA
SCHEMBL31009152 0.71 POLQ (0.41) ROCK2SCDSCN9ACACNA1BCACNA1C
SCHEMBL16895234 0.69 ROCK2 (0.40) ROCK2SCDSCN9A
SCHEMBL22462822 0.69 ROCK2 (0.41) ROCK2
SCHEMBL22462845 0.69 TGFBR1 (0.43) ROCK2STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed