SCHEMBL29315913

SCHEMBL29315913

O=C(O)Cc1c(-c2cn[nH]c2)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 8/20 0.39
ROCK2 O75116 7/20 0.39
RXRA P19793 4/20 0.38
RXRB P28702 4/20 0.38
RXRG P48443 4/20 0.38
GCGR P47871 1/20 0.38
EGLN1 Q9GZT9 1/20 0.37
AGBL2 Q5U5Z8 1/20 0.37
GPR17 Q13304 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
BLM P54132 1/20 0.36
PDK2 Q15119 1/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
MYLK4 Q86YV6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29315909 0.87 ROCK2 (0.46) ROCK1ROCK2
SCHEMBL29314121 0.78 POLQ (0.44) ROCK1ROCK2
SCHEMBL29316278 0.77 NPBWR1 (0.39) ROCK1ROCK2BLMPDK2
SCHEMBL29315915 0.72 ROCK2 (0.37) ROCK2RXRARXRBRXRGGCGR
SCHEMBL29316276 0.70 ROCK2 (0.39) ROCK1ROCK2RXRARXRBRXRG
SCHEMBL29315902 0.69 RXRA (0.44) RXRARXRBRXRGEGLN1AGBL2
SCHEMBL2996698 0.68 RXRA (0.50) ROCK1ROCK2RXRARXRBRXRG
SCHEMBL15245170 0.65 METAP2 (0.68)
SCHEMBL6864341 0.65 CES2 (0.46) RXRARXRBRXRGEGLN1GPR17
SCHEMBL20040983 0.64 NPBWR1 (0.44) ROCK1ROCK2PDK2MYLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed