SCHEMBL2931689

SCHEMBL2931689

COc1ccc(C=Cc2[c]cccc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.61
RELA Q04206 7/20 0.52
NFE2L2 Q16236 4/20 0.50
CYP1A2 P05177 3/20 0.50
CYP1A1 P04798 3/20 0.50
CYP1B1 Q16678 3/20 0.50
ESR1 P03372 2/20 0.50
PTGS2 P35354 2/20 0.50
ABL1 P00519 1/20 0.50
TTR P02766 1/20 0.50
ABCB1 P08183 1/20 0.50
ALOX5 P09917 1/20 0.50
BCR P11274 1/20 0.50
CYP19A1 P11511 1/20 0.50
NQO2 P16083 1/20 0.50
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
AHR P35869 1/20 0.50
TUBA1B P68363 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2938818 0.80 FGF23 (0.46) RELANFE2L2PTGS2ALOX5TUBB4A
SCHEMBL191091 0.79 CHAT (0.45) TRPA1RELANFE2L2ALOX5CYP19A1
SCHEMBL191092 0.79 CHAT (0.45) TRPA1RELANFE2L2ALOX5CYP19A1
SCHEMBL8591467 0.79 RELA (0.55) TRPA1RELANFE2L2CYP1A2CYP1A1
SCHEMBL699621 0.77 TRPA1 (1.00) TRPA1RELANFE2L2CYP1A2CYP1A1
SCHEMBL699620 0.77 TRPA1 (1.00) TRPA1RELANFE2L2CYP1A2CYP1A1
SCHEMBL8845585 0.77 TRPA1 (1.00) TRPA1RELANFE2L2CYP1A2CYP1A1
SCHEMBL7128336 0.77 AHR (0.60) TRPA1RELANFE2L2CYP1A2CYP1A1
SCHEMBL5664436 0.77
SCHEMBL631998 0.77 RELA (0.81) TRPA1RELANFE2L2CYP1A2CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1978967-B1 QUINAZOLINONE DERIVATIVES AS VANILLOID ANTAGONISTS NOVARTIS AG (CH) 2010-09-22 EP claimed
CN-108558927-B Silicon stereocenter chiral compound and synthesis method thereof 杭州师范大学 2020-06-19 CN disclosed
CN-108558927-A A kind of silicon Stereocenter chipal compounds and its synthetic method 杭州师范大学 2018-09-21 CN disclosed
EP-1978967-B1 QUINAZOLINONE DERIVATIVES AS VANILLOID ANTAGONISTS NOVARTIS AG (CH) 2010-09-22 EP disclosed