SCHEMBL2932836

SCHEMBL2932836

O=C(O)CNC(=O)c1ccc(Nc2cncc(-c3cc4ccccc4[nH]3)n2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITK Q08881 4/20 0.41
FTO Q9C0B1 5/20 0.41
EGLN1 Q9GZT9 5/20 0.41
HIF1AN Q9NWT6 4/20 0.41
KDM6B O15054 2/20 0.41
KDM5B Q9UGL1 2/20 0.41
KDM3A Q9Y4C1 1/20 0.41
EGFR P00533 2/20 0.40
PIK3CA P42336 2/20 0.40
BRAF P15056 1/20 0.40
DGAT1 O75907 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
BTK Q06187 1/20 0.38
IDO1 P14902 1/20 0.38
KDR P35968 1/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2934019 0.83 BRAF (0.47) ITKBRAF
Acetic Acid SCHEMBL2933253 0.82 BRAF (0.47) ITKEGFRPIK3CABRAF
SCHEMBL2933256 0.79 BRAF (0.57) ITKBRAF
SCHEMBL2927043 0.76 HCAR3 (0.48) ITKBRAF
SCHEMBL2928571 0.76 BTK (0.53) PIK3CABRAFBTKRAB9ASMN1; SMN2
SCHEMBL2931626 0.76 BRAF (0.39) ITKBRAFKDR
SCHEMBL2928708 0.76 BRAF (0.39) ITKBRAFKDR
Acetic Acid SCHEMBL2934985 0.75 BTK (0.52) PIK3CABRAFBTKRAB9ASMN1; SMN2
SCHEMBL27744978 0.75 BRAF (0.36) ITKBRAFKDR
SCHEMBL27745009 0.75 BRAF (0.36) ITKBRAFKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044051-B1 PYRIDINE AND PYRAZINE DERIVATIVES AS MNK KINASE INHIBITORS BIOVITRUM AB PUBL (SE) 2010-01-27 EP claimed