SCHEMBL29329720

SCHEMBL29329720

N#Cc1cc(Oc2cccc(C(F)(F)F)c2)cc(Nc2ccc3cc[nH]c3c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTBK1 Q5TCY1 2/20 0.46
TTBK2 Q6IQ55 1/20 0.46
ESR1 P03372 2/20 0.45
CDK8 P49336 2/20 0.40
IDH1 O75874 1/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
ERBB3 P21860 1/20 0.40
ERBB4 Q15303 1/20 0.40
KIF11 P52732 1/20 0.39
POLB P06746 1/20 0.38
CTSS P25774 1/20 0.37
PRKCQ Q04759 2/20 0.36
BRAF P15056 2/20 0.36
KDR P35968 1/20 0.36
P2RY1 P47900 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
NR3C1 P04150 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29330248 0.90 ESR1 (0.46) TTBK1TTBK2ESR1CDK8PRKCQ
SCHEMBL29330092 0.89 ABL1 (0.41) TTBK1TTBK2ESR1EGFRERBB2
SCHEMBL29330094 0.88 PRKCQ (0.40) TTBK1TTBK2ESR1CDK8PRKCQ
SCHEMBL29328747 0.86 EGFR (0.42) TTBK1TTBK2ESR1EGFRERBB2
SCHEMBL29330567 0.86 PRKCQ (0.45) TTBK1TTBK2ESR1POLBPRKCQ
SCHEMBL29329869 0.85 ESR1 (0.42) ESR1IDH1KIF11POLB
SCHEMBL29328660 0.85 SYK (0.39) ESR1PRKCQBRAFKDR
SCHEMBL29329538 0.85 SYK (0.39) ESR1CDK8EGFRPRKCQBRAF
SCHEMBL29329432 0.85 PRKCQ (0.38) TTBK1TTBK2ESR1EGFRERBB2
SCHEMBL29329642 0.84 ABL1 (0.46) TTBK1TTBK2ESR1CTSSPRKCQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024151919-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY IFM DUE, INC. (US) 2024-07-18 WO disclosed