SCHEMBL2933110

SCHEMBL2933110

OCC(F)(F)c1cc(Br)cs1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13759874 0.77 ALDH1A1 (0.37) CES2CES1ALDH1A1LMNAGSK3B
SCHEMBL20547211 0.77 CES2 (0.36) CES2CES1ALDH1A1LMNAGSK3B
SCHEMBL16621609 0.68 ALDH1A1 (0.34) CES2CES1ALDH1A1LMNAGSK3B
SCHEMBL2933069 0.68 CES2 (0.34) CES2CES1
SCHEMBL14415984 0.68 CES2 (0.34) CES2CES1ALDH1A1LMNAGSK3B
SCHEMBL10022930 0.67 CES2 (0.36) CES2CES1ALDH1A1LMNAGSK3B
SCHEMBL24917699 0.67
SCHEMBL15903198 0.66 CETP (0.31) ALDH1A1LMNA
SCHEMBL19134548 0.65 CES2 (0.31) CES2CES1ALDH1A1LMNAGSK3B
SCHEMBL16744594 0.64 PTGS2 (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229373-A1 SUBSTITUTED 2-NAPHTHOIC ACIDS AS ANTAGONISTS OF GPR105 ACTIVITY Merck Frosst Canada Ltd. (CA) 2010-09-22 EP disclosed
WO-2009070873-A1 SUBSTITUTED 2-NAPHTHOIC ACIDS AS ANTAGONISTS OF GPR105 ACTIVITY MERCK FROSST CANADA LTD. (CA) 2009-06-11 WO disclosed