SCHEMBL29337108

SCHEMBL29337108

C[C@@H](N)c1cccc(C#N)n1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.39
IDH1 O75874 1/20 0.38
IRAK4 Q9NWZ3 3/20 0.37
SOS2 Q07890 1/20 0.37
CTSS P25774 2/20 0.35
ADORA2A P29274 4/20 0.34
PARP1 P09874 1/20 0.33
IKBKB O14920 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31146070 1.00 CTSK (0.39) CTSKIDH1IRAK4SOS2CTSS
SCHEMBL22230336 1.00 CTSK (0.39) CTSKIDH1IRAK4SOS2CTSS
Hydrochloric Acid SCHEMBL22230342 0.98 CTSK (0.38) CTSKIDH1IRAK4SOS2CTSS
Hydrochloric Acid SCHEMBL22230340 0.98 CTSK (0.38) CTSKIDH1IRAK4SOS2CTSS
SCHEMBL179277 0.84 HSD11B1 (0.41) CTSKIDH1SOS2CTSSADORA2A
SCHEMBL20738618 0.81 IDH1 (0.38) CTSKIDH1SOS2CTSSADORA2A
SCHEMBL20989227 0.81 IDH1 (0.38) CTSKIDH1SOS2CTSSADORA2A
SCHEMBL17574520 0.80 CTSS (0.36) CTSKIDH1IRAK4SOS2CTSS
Hydrochloric Acid SCHEMBL1111090 0.79 TAAR1 (0.36) CTSKIDH1IRAK4SOS2CTSS
SCHEMBL522063 0.79 CYP1A2 (0.38) IRAK4ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3365334-B1 BENZOLACTAM COMPOUNDS AS PROTEIN KINASE INHIBITORS OTSUKA PHARMA CO LTD (JP) 2024-07-17 EP disclosed