SCHEMBL29338289

SCHEMBL29338289

COc1ccc2c(c1)CCN(C(=O)CN)CC2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.56
ESR2 Q92731 1/20 0.56
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA7 P43166 1/20 0.53
CA9 Q16790 1/20 0.53
CA14 Q9ULX7 1/20 0.53
DRD1 P21728 5/20 0.51
DRD5 P21918 5/20 0.51
DRD2 P14416 4/20 0.51
DRD3 P35462 4/20 0.51
ABHD6 Q9BV23 1/20 0.51
DRD4 P21917 2/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
TAAR1 Q96RJ0 1/20 0.49
NOTUM Q6P988 1/20 0.49
MEN1 O00255 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10351344 0.82 ESR1 (0.62) ESR1ESR2CA1CA2CA7
SCHEMBL11455526 0.81 KMT2A (0.66) ESR1ESR2DRD1DRD5DRD2
SCHEMBL3157287 0.81 ESR1 (0.52) ESR1ESR2CA1CA2CA7
SCHEMBL12209611 0.78 MTNR1B (0.60) ESR1ESR2CA1CA2CA7
SCHEMBL10400059 0.78 ESR1 (0.64) ESR1ESR2CA1CA2CA7
SCHEMBL29338249 0.78 SLC6A15 (0.54) NOTUMMEN1KMT2ASMN1; SMN2LMNA
SCHEMBL11457061 0.77 MTNR1B (0.64) ESR1ESR2CA1CA2CA7
SCHEMBL2309023 0.77 ESR1 (0.85) ESR1ESR2CA1CA2CA7
SCHEMBL3150165 0.77 RYR2 (0.58) ESR1ESR2CA1CA2CA7
SCHEMBL521554 0.77 KMT2A (0.48) MEN1KMT2AABCB1ABCC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3365334-B1 BENZOLACTAM COMPOUNDS AS PROTEIN KINASE INHIBITORS OTSUKA PHARMA CO LTD (JP) 2024-07-17 EP disclosed