SCHEMBL29338673

SCHEMBL29338673

Cc1cc(Br)cnc1CBr

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
ERBB2 P04626 1/20 0.36
HTT P42858 2/20 0.35
KMT2A Q03164 1/20 0.35
AGBL2 Q5U5Z8 2/20 0.34
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
DYRK1A Q13627 2/20 0.31
UHRF1 Q96T88 1/20 0.31
NPC1 O15118 1/20 0.31
GBA1 P04062 1/20 0.31
AAK1 Q2M2I8 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18489099 0.83 S1PR1 (0.35) S1PR1S1PR3SMN1; SMN2HTTKMT2A
SCHEMBL15080876 0.83 S1PR1 (0.37) S1PR1S1PR3SMN1; SMN2HTTKMT2A
SCHEMBL7751886 0.81 S1PR1 (0.39) S1PR1S1PR3SMN1; SMN2HTTKMT2A
SCHEMBL16809676 0.81 S1PR1 (0.39) S1PR1S1PR3SMN1; SMN2HTTKMT2A
SCHEMBL1577276 0.81 AGBL2 (0.37) S1PR1S1PR3SMN1; SMN2HTTKMT2A
SCHEMBL2112705 0.81 S1PR1 (0.39) S1PR1S1PR3SMN1; SMN2HTTKMT2A
SCHEMBL3392232 0.80 NOS3 (0.46) ERBB2AGBL2UHRF1CYP2A6
SCHEMBL17841682 0.78 AGXT (0.35) S1PR1S1PR3SMN1; SMN2HTTKMT2A
SCHEMBL5733354 0.78 S1PR1 (0.34) S1PR1S1PR3SMN1; SMN2HTTKMT2A
SCHEMBL7430667 0.78 S1PR1 (0.37) S1PR1S1PR3SMN1; SMN2HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3365334-B1 BENZOLACTAM COMPOUNDS AS PROTEIN KINASE INHIBITORS OTSUKA PHARMA CO LTD (JP) 2024-07-17 EP disclosed