SCHEMBL29355446

SCHEMBL29355446

CCCCOC(=O)Nc1ncc(C(O)c2cccc(OC)c2)s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.54
ALDH1A1 P00352 5/20 0.48
KDM4E B2RXH2 3/20 0.47
HPGD P15428 3/20 0.47
GAA P10253 2/20 0.47
HSD17B10 Q99714 2/20 0.46
SCD O00767 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
USP2 O75604 1/20 0.45
RAB9A P51151 4/20 0.45
NPC1 O15118 2/20 0.45
CYP1A2 P05177 1/20 0.45
NFKB1 P19838 1/20 0.45
CYP2C19 P33261 1/20 0.45
STAT1 P42224 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
CDK5 Q00535 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29358930 0.87 RAB9A (0.46) TSHRALDH1A1KDM4EHPGDGAA
SCHEMBL21384077 0.82 CCNE1 (0.49) ALDH1A1SCDSMN1; SMN2RAB9ANPC1
SCHEMBL21395005 0.82 CCNE1 (0.47) ALDH1A1KDM4EHPGDHSD17B10SCD
SCHEMBL29357987 0.82 CCNE1 (0.47) ALDH1A1KDM4EHPGDHSD17B10SCD
SCHEMBL29358368 0.75 L3MBTL1 (0.45) TSHRALDH1A1KDM4EHPGDGAA
SCHEMBL34467367 0.71 CDK2 (0.47) ALDH1A1SCDSMN1; SMN2CCNE1CDK2
SCHEMBL5502790 0.70 SMN1; SMN2 (0.47) TSHRGAASMN1; SMN2RAB9ANPC1
SCHEMBL2654505 0.70 L3MBTL1 (0.59) TSHRALDH1A1KDM4EHPGDGAA
SCHEMBL29353713 0.70 SMN1; SMN2 (0.64) TSHRALDH1A1KDM4EGAAHSD17B10
SCHEMBL29356285 0.70 TSHR (0.50) TSHRALDH1A1KDM4EHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3941908-A1 COMPOUNDS AND USES THEREOF Yumanity Therapeutics, Inc. (US) 2022-01-26 EP disclosed