SCHEMBL21395005

SCHEMBL21395005

COc1cccc(C(O)c2cnc(NC(=O)OC(C)(C)C)s2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 1/20 0.47
CDK2 P24941 1/20 0.47
CDK5 Q00535 1/20 0.47
SCD O00767 2/20 0.46
LCK P06239 2/20 0.41
GLS O94925 1/20 0.40
P2RY2 P41231 1/20 0.39
HSD17B10 Q99714 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
DYRK3 O43781 1/20 0.39
PRKCG P05129 1/20 0.39
PRKACA P17612 1/20 0.39
RPS6KB1 P23443 1/20 0.39
MAPK1 P28482 1/20 0.39
CLK2 P49760 1/20 0.39
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39
RPS6KA3 P51812 1/20 0.39
PRKCD Q05655 1/20 0.39
ROCK1 Q13464 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29357987 1.00 CCNE1 (0.47) CCNE1CDK2CDK5SCDLCK
SCHEMBL34467367 0.88 CDK2 (0.47) CCNE1CDK2CDK5SCDLCK
SCHEMBL21394890 0.86 S1PR3 (0.46) CCNE1CDK2CDK5SCDLCK
SCHEMBL21394898 0.86 SCD (0.45) CCNE1CDK2CDK5SCDLCK
SCHEMBL29356596 0.86 SCD (0.45) CCNE1CDK2CDK5SCDLCK
SCHEMBL29358752 0.86 S1PR3 (0.46) CCNE1CDK2CDK5SCDLCK
SCHEMBL21384077 0.85 CCNE1 (0.49) CCNE1CDK2CDK5SCDGLS
SCHEMBL29355446 0.82 TSHR (0.54) CCNE1CDK2CDK5SCDGLS
SCHEMBL21394896 0.81 P2RY2 (0.42) CCNE1CDK2CDK5SCDLCK
SCHEMBL21394886 0.79 P2RY2 (0.53) CCNE1CDK2CDK5P2RY2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed