Fevipiprant

Fevipiprant

SCHEMBL29355753

Cc1c(CC(=O)O)c2cccnc2n1Cc1ccc(S(C)(=O)=O)cc1C(F)(F)F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGDR2

The experimentally established mechanism targets of Fevipiprant. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PTGDR2 known ✓ Q9Y5Y4 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fevipiprant SCHEMBL1940595 1.00 PTGDR2 (1.00) PTGDR2
SCHEMBL1939556 0.92 PTGDR2 (1.00) PTGDR2
SCHEMBL21591931 0.90 PTGDR2 (0.82) PTGDR2
SCHEMBL1940778 0.90 PTGDR2 (0.82) PTGDR2
SCHEMBL20508235 0.90 PTGDR2 (0.81) PTGDR2
SCHEMBL21913709 0.89 PTGDR2 (0.80) PTGDR2
SCHEMBL1940435 0.88 PTGDR2 (1.00) PTGDR2
SCHEMBL1941189 0.87 PTGDR2 (1.00) PTGDR2
SCHEMBL1941253 0.87 PTGDR2 (0.82) PTGDR2
SCHEMBL28356397 0.87 PTGDR2 (0.76) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 224 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12533095-B1 Airway mucus scoring system THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-01-27 US claimed
WO-2025264860-A2 METHODS OF TREATING POST-COVID AIRWAY DISEASE YALE UNIVERSITY (US) 2025-12-26 WO claimed
US-20250381192-A1 Treatment of Autoimmune Disease JAK SLAVE PTY LTD (AU) 2025-12-18 US claimed
US-12364696-B2 Treatment of autoimmune disease JAK SLAVE PTY LTD (AU) 2025-07-22 US claimed
WO-2024192765-A1 FIRST IN CLASS USE OF THE CRTH2 ANTAGONIST IN TREATING NEUROMYELITIS OPTICA SPECTRUM DISORDER (NMOSD) AND RELEVANT AUTOIMMUNE CNS DISORDERS BROWN UNIVERSITY (US) 2024-09-26 WO claimed
US-12091708-B2 Compositions and methods targeting the Th2 pathway for the treatment of asthma THE CHILDREN'S HOSPITAL OF PHILADELPHIA (US) 2024-09-17 US claimed
US-20240226057-A1 NEW USE OF MONENSIN MAST PHARMA AB (SE) 2024-07-11 US claimed
EP-4378957-A2 COMBINATION THERAPIES COMPRISING ANTIBODY MOLECULES TO PD-1 Novartis AG (CH) 2024-06-05 EP claimed
US-20240148745-A1 COMPOUNDS FOR USE IN PROGRESSIVE MULTIPLE SCLEROSIS FONDAZIONE CENTRO SAN RAFFAELE (IT) 2024-05-09 US claimed
EP-4362934-A1 NEW USE OF MONENSIN Mast Pharma AB (SE) 2024-05-08 EP claimed
CN-117612741-A Novel coronavirus infection metabolic profile, and construction method, device, system and application thereof 首都医科大学附属北京朝阳医院 2024-02-27 CN claimed
EP-4304719-A1 COMPOUNDS FOR USE IN PROGRESSIVE MULTIPLE SCLEROSIS Fondazione Centro San Raffaele (IT) 2024-01-17 EP claimed
WO-2023277761-A1 NEW USE OF MONENSIN PEJLER GUNNAR (SE) 2023-01-05 WO claimed
WO-2022189531-A1 COMPOUNDS FOR USE IN PROGRESSIVE MULTIPLE SCLEROSIS FONDAZIONE CENTRO SAN RAFFAELE (IT) 2022-09-15 WO claimed
EP-4056231-A1 COMPOUNDS FOR USE IN PROGRESSIVE MULTIPLE SCLEROSIS Fondazione Centro San Raffaele (IT) 2022-09-14 EP claimed
US-20220259656-A1 BLOOD BIOMARKER AND GENETIC MARKERS ASSOCIATED WITH RESPONSE TO CRTH2 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2022-08-18 US claimed
EP-3337803-B1 GENETIC MARKERS ASSOCIATED WITH RESPONSE TO CRTH2 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LLC (US) 2022-08-17 EP claimed
US-20220187316-A1 Postural Orthostatic Tachycardia Syndrome and CRTH2 AMERIMMUNE DIAGNOSTICS LLC 2022-06-16 US claimed
US-20220143025-A1 TREATMENT OF AUTOIMMUNE DISEASE JAK SLAVE PTY LTD (AU) 2022-05-12 US claimed
EP-3941579-A1 POSTURAL ORTHOSTATIC TACHYCARDIA SYNDROME AND CRTH2 Amerimmune, LLC (US) 2022-01-26 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12364696-B2 Treatment of autoimmune disease JAK1, JAK3, JAK2 PTGDR2 2062/4885
US-20250381192-A1 Treatment of Autoimmune Disease JAK1, JAK3, JAK2 PTGDR2 2062/4885
US-20220143025-A1 TREATMENT OF AUTOIMMUNE DISEASE JAK1, JAK3, JAK2 PTGDR2 2062/4885
US-20240226057-A1 NEW USE OF MONENSIN MRGPRX1, MRGPRX2, CMA1 PTGDR2 1558/4885
US-12533095-B1 Airway mucus scoring system MUC1, IL5, CYSLTR2 PTGDR2 637/4885
US-20220259656-A1 BLOOD BIOMARKER AND GENETIC MARKERS ASSOCIATED WITH RESPONSE TO CRTH2 RECEPTOR ANTAGONISTS HRH2, HRH1, CRHR2 PTGDR2 28/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.