SCHEMBL29360910

SCHEMBL29360910

COC(=O)[C@H](Cc1ccc(Cl)cc1)NC(=O)c1cc2cc(Cl)ccc2[nH]1

nearest known ligand 0.88

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PYGL P06737 11/20 0.88
CYP51A1 Q16850 6/20 0.64
CTNNB1 P35222 1/20 0.62
EGFR P00533 1/20 0.59
PYGM P11217 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165218 0.94 PYGL (0.81) PYGLCYP51A1CTNNB1EGFRPYGM
SCHEMBL29362778 0.94 PYGL (0.81) PYGLCYP51A1CTNNB1EGFRPYGM
SCHEMBL6165213 0.94 PYGL (0.81) PYGLCYP51A1CTNNB1EGFRPYGM
SCHEMBL14587604 0.94 PYGL (1.00) PYGLCYP51A1CTNNB1EGFR
SCHEMBL6161267 0.94 PYGL (1.00) PYGLCYP51A1CTNNB1EGFR
SCHEMBL29357801 0.92 PYGL (0.78) PYGLCYP51A1CTNNB1EGFRPYGM
SCHEMBL29359765 0.91 PYGL (0.77) PYGLCYP51A1CTNNB1EGFRPYGM
SCHEMBL29359826 0.91 PYGL (0.77) PYGLCYP51A1CTNNB1EGFRPYGM
SCHEMBL29358053 0.90 PYGL (0.81) PYGLCTNNB1
SCHEMBL6163437 0.87 PYGL (0.74) PYGLCYP51A1CTNNB1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250289848-A1 PEPTIDOMIMETIC INHIBITORS OF B-CATENIN/TCF PROTEIN-PROTEIN INTERACTION H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. 2025-09-18 US disclosed
US-12269899-B2 Peptidomimetic inhibitors of β-catenin/Tcf protein-protein interaction H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2025-04-08 US disclosed
US-20220024977-A1 PEPTIDOMIMETIC INHIBITORS OF B-CATENIN/TCF PROTEIN-PROTEIN INTERACTION H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. 2022-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250289848-A1 PEPTIDOMIMETIC INHIBITORS OF B-CATENIN/TCF PROTEIN-PROTEIN INTERACTION CTNNB1, CTNNBL1, CTNND1 PYGL 184/4885CYP51A1 780/4885CTNNB1 1/4885
US-12269899-B2 Peptidomimetic inhibitors of β-catenin/Tcf protein-protein interaction CTNNB1, CTNNBL1, CTNND1 PYGL 186/4885CYP51A1 695/4885CTNNB1 1/4885
US-20220024977-A1 PEPTIDOMIMETIC INHIBITORS OF B-CATENIN/TCF PROTEIN-PROTEIN INTERACTION CTNNB1, CTNNBL1, CTNND1 PYGL 184/4885CYP51A1 780/4885CTNNB1 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.