SCHEMBL29368281

SCHEMBL29368281

CC(C)(C)c1ccc(-c2cnc(C(=O)O)c(N)n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.47
ASIC3 Q9UHC3 1/20 0.45
COPS5 Q92905 3/20 0.45
DGAT1 O75907 1/20 0.43
ATR Q13535 8/20 0.43
PRKDC P78527 4/20 0.43
ATM Q13315 2/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ADORA2A P29274 1/20 0.41
LDHA P00338 1/20 0.41
LDHB P07195 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22712451 1.00 IKBKB (0.47) IKBKBASIC3COPS5DGAT1ATR
SCHEMBL22712516 0.85 IKBKB (0.44) IKBKBASIC3DGAT1ATRPRKDC
SCHEMBL29410008 0.85 IKBKB (0.44) IKBKBASIC3DGAT1ATRPRKDC
SCHEMBL319167 0.83 ASIC3 (0.57) IKBKBASIC3ATRPRKDCATM
SCHEMBL28175377 0.79 DGAT1 (0.51) IKBKBDGAT1PRKDCNPC1RAB9A
SCHEMBL23703565 0.75 PIK3CD (0.53) ATRPRKDCATM
SCHEMBL22732755 0.73 DGAT1 (0.45) IKBKBDGAT1PRKDCNPC1RAB9A
SCHEMBL30048631 0.73 ATR (0.67) ATRPRKDCATM
SCHEMBL23703073 0.73 ATR (0.67) ATRPRKDCATM
SCHEMBL26941761 0.73 DGAT1 (0.45) DGAT1PRKDCNPC1RAB9AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115215923-B Macrocyclic broad-spectrum antibiotics 豪夫迈·罗氏有限公司 2026-05-19 CN disclosed
CN-115215923-A Macrocyclic broad spectrum antibiotics 豪夫迈·罗氏有限公司 2022-10-21 CN disclosed
CN-114007605-B Macrocyclic broad spectrum antibiotics 豪夫迈·罗氏有限公司 2022-07-15 CN disclosed
EP-3968983-A1 MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS F. Hoffmann-La Roche AG (CH) 2022-03-23 EP disclosed
CN-114007605-A Macrocyclic broad spectrum antibiotics 豪夫迈·罗氏有限公司 2022-02-01 CN disclosed