SCHEMBL319167

SCHEMBL319167

Nc1nc(-c2ccccc2)cnc1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 1/20 0.57
ATR Q13535 10/20 0.56
PRKDC P78527 4/20 0.56
IKBKB O14920 1/20 0.50
ATM Q13315 2/20 0.48
CYP3A4 P08684 1/20 0.47
NEK2 P51955 1/20 0.47
NOS1 P29475 1/20 0.47
MAP2K3 P46734 1/20 0.46
LDHA P00338 1/20 0.46
TLR9 Q9NR96 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28324236 0.87 IKBKB (0.58) ASIC3ATRPRKDCIKBKBATM
SCHEMBL318797 0.86 ATR (0.68) ATRPRKDCIKBKBATMCYP3A4
SCHEMBL6987949 0.84 IKBKB (0.51) ASIC3ATRPRKDCIKBKBATM
SCHEMBL22712451 0.83 IKBKB (0.47) ASIC3ATRPRKDCIKBKBATM
SCHEMBL29368281 0.83 IKBKB (0.47) ASIC3ATRPRKDCIKBKBATM
SCHEMBL336653 0.83 ATR (0.53) ASIC3ATRPRKDCIKBKBATM
SCHEMBL26986900 0.81 IKBKB (0.48) ASIC3ATRPRKDCIKBKBLDHA
SCHEMBL28918651 0.79 ALDH1A1 (0.56) ATRPRKDCIKBKBLDHA
SCHEMBL5684569 0.79 ATR (0.63) ATRPRKDCATMCYP3A4
SCHEMBL24248259 0.78 ATR (0.67) ATRPRKDCIKBKBATMCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889683-B2 Substituted quinoxalines as inhibitors of fatty acid binding protein MERCK SHARP & DOHME CORP. (US) 2014-11-18 US disclosed
US-8889683-B2 Substituted quinoxalines as inhibitors of fatty acid binding protein MERCK SHARP & DOHME CORP. (US) 2014-11-18 US disclosed
EP-2590968-A1 CYCLIC ETHER COMPOUNDS USEFUL AS KINASE INHIBITORS Novartis AG (CH) 2013-05-15 EP disclosed
US-20120122837-A1 INHIBITORS OF FATTY ACID BINDING PROTEIN MERCK SHARP & DOHME LLC 2012-05-17 US disclosed
US-20120122837-A1 INHIBITORS OF FATTY ACID BINDING PROTEIN MERCK SHARP & DOHME LLC 2012-05-17 US disclosed
WO-2012004217-A1 CYCLIC ETHER COMPOUNDS USEFUL AS KINASE INHIBITORS NOVARTIS AG (CH) 2012-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122837-A1 INHIBITORS OF FATTY ACID BINDING PROTEIN FABP4, FABP1, FABP3 ASIC3 2273/4885ATR 4853/4885PRKDC 4822/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.