SCHEMBL29370504

SCHEMBL29370504

CCOC(=O)CC(NC1[C@H]2CN(C(=O)CCc3ccc4c(n3)N(C(=O)O)CCC4)C[C@@H]12)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
ITGB3 P05106 14/20 0.35
ITGAV P06756 14/20 0.35
ITGA2B P08514 8/20 0.35
ITGB5 P18084 7/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GRM7 Q14831 2/20 0.34
NPC1 O15118 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
ITGB6 P18564 1/20 0.34
ITGB8 P26012 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29392180 0.91 LMNA (0.36) LMNAITGB3ITGAVITGA2BITGB5
SCHEMBL29369724 0.89 LMNA (0.40) LMNAITGB3ITGAVITGB5ALDH1A1
SCHEMBL29370435 0.82 ITGB3 (0.37) LMNAITGB3ITGAVITGA2BITGB5
SCHEMBL29393359 0.81 LMNA (0.37) LMNAITGB3ITGAVITGB5ITGB6
Trifluoroacetic Acid SCHEMBL29393937 0.80 ITGB3 (0.48) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL20140313 0.78 NOTUM (0.40) ALDH1A1HPGDSMN1; SMN2
SCHEMBL21329619 0.74 BRD4 (0.39) ITGAVHPGDSMN1; SMN2ITGB6
SCHEMBL28708231 0.74 ITGB3 (0.37) ITGB3ITGAVITGA2BITGB5GRM7
SCHEMBL29390969 0.74 ITGAV (0.34) LMNAITGB3ITGAVITGB5ALDH1A1
SCHEMBL28694811 0.74 ITGB3 (0.36) LMNAITGB3ITGAVITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022022364-A1 PYRROLIDINE INTEGRIN MODULATOR AND USE THEREOF 清药同创(北京)药物研发中心有限公司 2022-02-03 WO disclosed