SCHEMBL28708231

SCHEMBL28708231

COC(=O)C(c1ccccc1)N(C)C1CCN(C(=O)CCc2ccc3c(n2)N(C(=O)O)CCC3)C1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 15/20 0.37
ITGAV P06756 15/20 0.37
ITGA2B P08514 11/20 0.37
ITGB5 P18084 8/20 0.36
ITGB1 P05556 1/20 0.35
KDM1A O60341 2/20 0.34
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
GRM7 Q14831 1/20 0.34
C3AR1 Q16581 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28692098 0.86 CCR5 (0.36) ITGAV
SCHEMBL30474545 0.85 ITGB3 (0.53) ITGB3ITGAVITGA2BITGB5ITGB1
SCHEMBL28699772 0.85 ITGB3 (0.53) ITGB3ITGAVITGA2BITGB5ITGB1
SCHEMBL28699770 0.85 ITGB3 (0.53) ITGB3ITGAVITGA2BITGB5ITGB1
SCHEMBL29370436 0.79 ITGAV (0.33) ITGB3ITGAVITGB5ITGB1
SCHEMBL28696946 0.78 CCR5 (0.39) ITGB3ITGAVITGB5
SCHEMBL28709388 0.77 ITGB3 (0.56) ITGB3ITGAVITGA2BITGB5ITGB1
SCHEMBL28709389 0.77 ITGB3 (0.56) ITGB3ITGAVITGA2BITGB5ITGB1
SCHEMBL28698380 0.75 KMT2A (0.40) KDM1AMAOAMAOB
SCHEMBL29370504 0.74 LMNA (0.39) ITGB3ITGAVITGA2BITGB5GRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed