SCHEMBL29370567

SCHEMBL29370567

CC(C)(CNC(=O)c1cccc(-c2noc(C(F)(F)F)n2)c1)c1coc(-c2ccccc2)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 15/20 1.00
HDAC1 Q13547 6/20 1.00
HDAC8 Q9BY41 5/20 1.00
HDAC7 Q8WUI4 4/20 1.00
HDAC5 Q9UQL6 4/20 1.00
HDAC9 Q9UKV0 3/20 1.00
HDAC6 Q9UBN7 13/20 0.49
HDAC3 O15379 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HPGDS O60760 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2226518 1.00 HDAC4 (1.00) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL2225769 0.94 HDAC4 (0.89) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL29757316 0.94 HDAC4 (0.88) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL2226555 0.93 HDAC4 (0.87) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL14605297 0.91 HDAC4 (0.82) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL14752448 0.88 HDAC4 (0.79) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL2228678 0.86 HDAC4 (0.76) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL2362796 0.83 HDAC4 (0.71) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL25049598 0.83 HDAC8 (0.71) HDAC4HDAC1HDAC8HDAC7HDAC5
SCHEMBL14752493 0.83 HDAC4 (0.71) HDAC4HDAC1HDAC8HDAC7HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 220 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
EP-4720316-A2 NON-VIRAL CELL ENGINEERING Arsenal Biosciences, Inc. (US) 2026-04-08 EP claimed
US-20250177529-A1 ACOUSTIC ENRICHMENT OF ADOPTIVE CELL TRANSFERS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE 2025-06-05 US claimed
US-20250144056-A1 ANTIMICROBIAL HOST DEFENSE PEPTIDE-INDUCING COMPOSITIONS AND METHODS OF PRODUCTION AND USE THEREOF BOARD OF REGENTS FOR THE OKLAHOMA AGRICULTURAL AND MECH COLLEGES (US) 2025-05-08 US claimed
US-20250115871-A1 METHODS TO IMPROVE ENDURING HEMATOPOIETIC STEM CELL TRANSPLANTATION TRAILHEAD BIOSYSTEMS INC. 2025-04-10 US claimed
US-20250090473-A1 Macrophage Targeted Immunotherapeutics THE GENERAL HOSPITAL CORPORATION 2025-03-20 US claimed
WO-2025059442-A1 MODULATING PLANT RESPONSES TO STRESS AND GROWTH WITH CHEMICALS REMOTE EPIGENETICS INC. (US) 2025-03-20 WO claimed
WO-2024259376-A2 NON-VIRAL CELL ENGINEERING ARSENAL BIOSCIENCES, INC. (US) 2024-12-19 WO claimed
US-20240366784-A1 INJECTABLE HYDROGEL COMPOSITIONS AND METHODS OF USE THEREOF DREXEL UNIVERSITY 2024-11-07 US claimed
US-20240358767-A1 STEM CELL DIFFERENTIATION AND CHEMICAL COMPOUNDS VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-10-31 US claimed
WO-2023167842-A2 ACOUSTIC ENRICHMENT OF ADOPTIVE CELL TRANSFERS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2023-09-07 WO claimed
WO-2023147573-A2 ANTIMICROBIAL HOST DEFENSE PEPTIDE-INDUCING COMPOSITIONS AND METHODS OF PRODUCTION AND USE THEREOF BOARD OF REGENTS FOR THE OKLAHOMA AGRICULTURAL AND MECHANICAL COLLEGES (US) 2023-08-03 WO claimed
CN-116510024-A Composition, preparation method and application thereof 上海复东生物医药有限责任公司 2023-08-01 CN claimed
WO-2023101943-A1 METHODS AND COMPOSITIONS FOR MAINTAINING AND EXPANDING HEMATOPOIETIC STEM CELLS TRAILHEAD BIOSYSTEMS INC. (US) 2023-06-08 WO claimed
WO-2023081884-A2 STEM CELL DIFFERENTIATION AND CHEMICAL COMPOUNDS VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-05-11 WO claimed
WO-2023074794-A1 METHOD OR AGENT WITH HDAC REGULATOR, FOR TREATMENT OF DIABETES AND COMPLICATIONS 国立大学法人滋賀医科大学 2023-05-04 WO claimed
CN-115778950-A Application of histone deacetylase inhibitor TMP195 in preparation of medicines for promoting osteogenesis 山西医科大学第二医院 2023-03-14 CN claimed
US-20230039816-A1 METHOD FOR INDUCING HEPATOCYTE PLASTICITY PUBLIC UNIVERSITY CORPORATION YOKOHAMA CITY UNIVERSITY (JP) 2023-02-09 US claimed
WO-2022192300-A1 STEM CELL DIFFERENTIATION AND POLYMERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-09-15 WO claimed
CN-115040660-A Mannitol modified nanoparticle and preparation method and application thereof 南通大学 2022-09-13 CN claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250090473-A1 Macrophage Targeted Immunotherapeutics CD47, CAPG, CD74 HDAC4 705/4885HDAC1 543/4885HDAC8 834/4885
US-20240366784-A1 INJECTABLE HYDROGEL COMPOSITIONS AND METHODS OF USE THEREOF CD44, PLOD3, TP53 HDAC4 3391/4885HDAC1 3551/4885HDAC8 2257/4885
US-20240358767-A1 STEM CELL DIFFERENTIATION AND CHEMICAL COMPOUNDS EBP, AKT3, PRKCD HDAC4 1053/4885HDAC1 512/4885HDAC8 1340/4885
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES WNT3A, GSK3B, GSK3A HDAC4 27/4885HDAC1 71/4885HDAC8 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.