SCHEMBL29375692

SCHEMBL29375692

OC(O)C1NCCc2c1[nH]c1ccccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C19 P33261 1/20 0.60
MAPKAPK2 P49137 1/20 0.59
GRIN2B Q13224 1/20 0.55
DRD2 P14416 1/20 0.54
HTR2A P28223 3/20 0.50
HTR2C P28335 3/20 0.50
KDM4E B2RXH2 1/20 0.50
HTR5A P47898 1/20 0.50
NISCH Q9Y2I1 1/20 0.50
NR2E1 Q9Y466 1/20 0.50
BRD3 Q15059 1/20 0.50
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PRMT5 O14744 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21326157 0.85 HTR7 (0.60) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
SCHEMBL18669403 0.80 HTR7 (0.58) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
SCHEMBL10814283 0.79 HTR7 (0.53) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
Tetrahydroharman SCHEMBL7018798 0.76 HTR7 (0.65) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
Tetrahydroharman SCHEMBL21012020 0.76 HTR7 (0.65) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
SCHEMBL12212162 0.76 HTR7 (0.65) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
Tetrahydroharman SCHEMBL29630296 0.76 HTR7 (0.65) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
SCHEMBL968830 0.76 HTR7 (0.65) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
SCHEMBL17839824 0.76 HTR7 (0.65) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2
Tetrahydroharman SCHEMBL29630308 0.76 HTR7 (0.65) HTR7CYP3A4CYP2D6CYP2C19MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109134605-B 1, 1-dihydroxymethyl-tetrahydro-beta-carboline-3-formyl-GYIGSK, and synthesis, activity and application thereof 首都医科大学 2022-04-22 CN claimed
CN-109134604-B 1, 1-dihydroxymethyl-tetrahydro-beta-carboline-3-formyl-GRGDF, and synthesis, activity and application thereof 首都医科大学 2022-04-22 CN claimed
CN-109111502-B 1, 1-dihydroxymethyl-tetrahydro-beta-carboline-3-formyl-GGPRP, and synthesis, activity and application thereof 首都医科大学 2022-04-22 CN claimed
CN-109134603-B 1, 1-dihydroxymethyl-tetrahydro-beta-carboline-3-formyl-GYIGSR, and synthesis, activity and application thereof 首都医科大学 2022-04-22 CN claimed
CN-109134607-B 1, 1-dihydroxymethyl-tetrahydro-beta-carboline-3-formyl-GRGDS, synthesis, activity and application thereof 首都医科大学 2022-02-08 CN claimed
CN-109134606-B 1, 1-dihydroxymethyl-tetrahydro-beta-carboline-3-formyl-GRGDV, synthesis, activity and application thereof 首都医科大学 2022-02-08 CN claimed