SCHEMBL2938806

SCHEMBL2938806

O=c1[nH]cnc2c1ccc1ncccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.56
PDPK1 O15530 1/20 0.56
CA12 O43570 1/20 0.56
ALOX15 P16050 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
CA9 Q16790 1/20 0.56
TNKS2 Q9H2K2 1/20 0.56
ACVR1 Q04771 4/20 0.56
PIM1 P11309 2/20 0.54
AURKA O14965 1/20 0.54
DAPK3 O43293 1/20 0.54
JAK2 O60674 1/20 0.54
PRKD3 O94806 1/20 0.54
MAP4K4 O95819 1/20 0.54
PAK4 O96013 1/20 0.54
ABL1 P00519 1/20 0.54
CSF1R P07333 1/20 0.54
RET P07949 1/20 0.54
IGF1R P08069 1/20 0.54
MET P08581 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31322342 0.78 PARP1 (0.68) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL2015165 0.77 LMNA (0.56) PARP1PDPK1CA12ALOX15SMN1; SMN2
Samoquasine A SCHEMBL15954512 0.76 PARP1 (0.57) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL30482888 0.76 LMNA (0.55) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL349009 0.73 PARP1 (0.55) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL334691 0.73 PARP1 (0.55) PARP1PDPK1CA12ALOX15SMN1; SMN2
Quinazolinone SCHEMBL27983253 0.72 PARP1 (1.00) PARP1PDPK1CA12ALOX15SMN1; SMN2
Quinazolinone SCHEMBL88525 0.72 PARP1 (1.00) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL12068009 0.72 PARP1 (0.66) PARP1PDPK1CA12ALOX15SMN1; SMN2
SCHEMBL29130935 0.72 PARP1 (0.53) PARP1PDPK1CA12ALOX15SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1978967-B1 QUINAZOLINONE DERIVATIVES AS VANILLOID ANTAGONISTS NOVARTIS AG (CH) 2010-09-22 EP claimed
EP-1978967-B1 QUINAZOLINONE DERIVATIVES AS VANILLOID ANTAGONISTS NOVARTIS AG (CH) 2010-09-22 EP disclosed