SCHEMBL29404479

SCHEMBL29404479

NC(N)=NCCC[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
MEN1 O00255 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
KMT2A Q03164 1/20 0.56
TPSAB1 Q15661 3/20 0.48
SIRT2 Q8IXJ6 2/20 0.47
SIRT1 Q96EB6 2/20 0.47
MME P08473 1/20 0.46
ECE1 P42892 1/20 0.46
CTSB P07858 3/20 0.45
CTSK P43235 3/20 0.45
ITGB3 P05106 2/20 0.45
ITGA2B P08514 2/20 0.45
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
AR P10275 1/20 0.43
MAP2K1 Q02750 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29918749 0.91 ALDH1A1 (0.49) KDM4EMEN1ALDH1A1LMNAHPGD
SCHEMBL29601597 0.89 SIRT2 (0.51) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL20660119 0.89 SIRT2 (0.51) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL7541299 0.88 KDM4E (0.56) KDM4EMEN1ALDH1A1LMNAHPGD
SCHEMBL29357202 0.87 SIRT1 (0.53) KDM4EALDH1A1HPGDTPSAB1SIRT2
SCHEMBL30141948 0.86 SIRT2 (0.49) KDM4EMEN1ALDH1A1LMNAHPGD
SCHEMBL29791017 0.86 SIRT2 (0.49) KDM4EMEN1ALDH1A1LMNAHPGD
SCHEMBL7740151 0.86 KDM4E (0.59) KDM4EMEN1ALDH1A1LMNAHPGD
Hydrochloric Acid SCHEMBL22413023 0.86 SIRT2 (0.48) TPSAB1SIRT2SIRT1MMEECE1
Hydrochloric Acid SCHEMBL31755364 0.86 SIRT2 (0.48) TPSAB1SIRT2SIRT1MMEECE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024197174-A1 PEPTIDE SUBSTRATES AND INHIBITORS OF CATHEPSIN B THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-09-26 WO disclosed
WO-2024030500-A1 COMPOSITIONS AND METHODS FOR TREATING PANCREATITIS GUKOVSKAYA ANNA (US) 2024-02-08 WO disclosed
EP-4294802-A1 CRYPTOPHYCIN COMPOUNDS AND CONJUGATES THEREOF Universität Bielefeld (DE) 2023-12-27 EP disclosed
WO-2022175222-A1 CRYPTOPHYCIN COMPOUNDS AND CONJUGATES THEREOF UNIVERSITÄT BIELEFELD (DE) 2022-08-25 WO disclosed
CN-114177199-A Polypeptide-modified gold cluster and application of polypeptide-modified gold cluster in resisting tumor invasion and metastasis by inhibiting activity of cathepsin B 北京工业大学 2022-03-15 CN disclosed