SCHEMBL29409999

SCHEMBL29409999

COCOc1cc(C(C)(C)C)ccc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.43
HIF1A Q16665 1/20 0.36
DGAT1 O75907 1/20 0.32
KDM4E B2RXH2 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CYP2C19 P33261 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22712518 1.00 EGFR (0.43) EGFRHIF1ADGAT1KDM4ECA1
SCHEMBL29276144 0.88 LIPE (0.36) EGFRKDM4EALDH1A1HTTCYP2C19
SCHEMBL26601625 0.88 MAPT (0.37) EGFRHIF1ADGAT1KDM4EALDH1A1
SCHEMBL12118481 0.84 EGFR (0.36) EGFRHIF1ACA1CA2CA9
SCHEMBL19087000 0.82 CSF1R (0.34) EGFRHIF1AALDH1A1CYP2C19MAPT
SCHEMBL28544224 0.81 CA1 (0.31) EGFRHIF1ACA1CA2CA9
SCHEMBL21410221 0.81 EGFR (0.39) EGFR
SCHEMBL30973537 0.81 EGFR (0.39) EGFR
SCHEMBL2280832 0.81 SNCA (0.38) EGFRHIF1AKDM4ECA1CA2
SCHEMBL31652177 0.81 LPL (0.40) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007605-B Macrocyclic broad spectrum antibiotics 豪夫迈·罗氏有限公司 2022-07-15 CN disclosed
EP-3968983-A1 MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS F. Hoffmann-La Roche AG (CH) 2022-03-23 EP disclosed