Ergotamine

Ergotamine

SCHEMBL29420131

CN1C[C@H](C(=O)N[C@]2(C)O[C@@]3(O)[C@@H]4CCCN4C(=O)[C@H](Cc4ccccc4)N3C2=O)C=C2c3cccc4[nH]cc(c34)C[C@H]21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CHTR1D

The experimentally established mechanism targets of Ergotamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A known ✓ P08913 5/20 1.00
ADRA2B known ✓ P18089 5/20 1.00
ADRA2C known ✓ P18825 5/20 1.00
ADRA1D known ✓ P25100 4/20 1.00
ADRA1A known ✓ P35348 3/20 1.00
HTR1D known ✓ P28221 1/20 1.00
ADRA1B known ✓ P35368 2/20 0.69
CYP3A4 P08684 9/20 1.00
DRD2 P14416 6/20 1.00
HTR2A P28223 6/20 1.00
HTR2C P28335 6/20 1.00
HTR6 P50406 6/20 1.00
HIF1A Q16665 5/20 1.00
DRD3 P35462 5/20 1.00
ABCB1 P08183 4/20 1.00
DRD1 P21728 4/20 1.00
HTR2B P41595 4/20 1.00
HTR1A P08908 4/20 1.00
CYP1A2 P05177 3/20 1.00
HTR1B P28222 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ergotamine SCHEMBL783018 1.00 CYP3A4 (1.00) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL22171508 1.00 CYP3A4 (1.00) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL18134607 1.00 CYP3A4 (1.00) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL1483 1.00 CYP3A4 (1.00) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL783017 1.00 CYP3A4 (1.00) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL453882 1.00 CYP3A4 (1.00) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL29567350 1.00 CYP3A4 (1.00) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL11086376 0.99 CYP3A4 (0.99) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL28990226 0.99 CYP3A4 (0.99) CYP3A4DRD2HTR2AHTR2CHTR6
Ergotamine SCHEMBL22231343 0.99 CYP3A4 (0.99) CYP3A4DRD2HTR2AHTR2CHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260071243-A1 BIOLOGICAL PRODUCTION OF TRYPTOPHAN-DERIVED PRODUCTS UNIV TEXAS (US) 2026-03-12 US disclosed
WO-2025226786-A1 METHODS AND COMPOSITIONS COMPRISING WETTABLE ELECTROSPUN MATRIX POLY-MED, INC. (US) 2025-10-30 WO disclosed
US-20250289909-A1 FUNCTIONALIZED AND CROSSLINKED POLYMERS PMIDG LLC (US) 2025-09-18 US disclosed
US-12351656-B2 Functionalized and crosslinked polymers PMIDG, LLC (US) 2025-07-08 US disclosed
US-20250161539-A1 INJECTION OF COLLAGEN ELASTIN HYDROGEL MICROPARTICLES INTO TORN TENDONS AND LIGAMENTS PETVIVO HOLDINGS INC (US) 2025-05-22 US disclosed
US-12303520-B2 Aqueous nebulization composition NEPHRON PHARMACEUTICALS CORPORATION (US) 2025-05-20 US disclosed
US-20250000693-A1 COMPOSITIONS, SYSTEMS AND METHODS FOR TREATING SUPRAPUBIC FAT MIRAKI INNOVATION THINK TANK LLC (US) 2025-01-02 US disclosed
WO-2024254456-A1 POINT OF USE DEVICE COATING PMIDG, LLC (US) 2024-12-12 WO disclosed
CN-118731222-A Extraction method and detection method of ergot alkaloid mycotoxins in pasture 呼和浩特海关技术中心 2024-10-01 CN disclosed
US-20240285517-A1 Biocompatible Protein-Based Particles and Methods Thereof PETVIVO HOLDINGS, INC. (US) 2024-08-29 US disclosed
EP-4121169-A2 INJECTABLE BOTULINUM TOXIN METHODS FOR TREATING HEADACHES ReVance Therapeutics, Inc. (US) 2023-01-25 EP disclosed
WO-2023278891-A1 COMPOSITIONS, SYSTEMS AND METHODS FOR TREATING SUPRAPUBIC FAT MIRAKI INNOVATION THINK TANK LLC (US) 2023-01-05 WO disclosed
US-20220296866-A1 METHODS, DEVICES AND COMPOSITIONS FOR LOCAL DELIVERY POLY-MED, INC. 2022-09-22 US disclosed
US-20220288092-A1 Aqueous Nebulization Composition NEPHRON PHARMACEUTICALS CORPORATION (US) 2022-09-15 US disclosed
US-11440976-B2 Functionalized and crosslinked polymers PMIDG, LLC (US) 2022-09-13 US disclosed
US-20220202703-A1 IN SITU GEL-FORMING DELIVERY SYSTEMS, METHODS AND COMPOSITIONS POLY-MED, INC. 2022-06-30 US disclosed
WO-2022120097-A1 FUNCTIONALIZED AND CROSSLINKED POLYMERS PMIDG, LLC (US) 2022-06-09 WO disclosed
US-11344562-B2 Aqueous nebulization composition NEPHRON PHARMACEUTICALS CORPORATION (US) 2022-05-31 US disclosed
EP-3979947-A1 METHODS, DEVICES AND COMPOSITIONS FOR LOCAL DELIVERY Poly-Med Inc. (US) 2022-04-13 EP disclosed
WO-2022032111-A1 ICED-WATER SLURRY FOR TREATING BROWN AND BEIGE FAT MIRAKI INNOVATION THINK TANK LLC (US) 2022-02-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11344562-B2 Aqueous nebulization composition PDE12, CYP11B2, IL5 ADRA2A 270/4885ADRA2B 81/4885ADRA2C 31/4885
US-20220288092-A1 Aqueous Nebulization Composition PDE12, CYP11B2, IL5 ADRA2A 270/4885ADRA2B 81/4885ADRA2C 31/4885
US-20260071243-A1 BIOLOGICAL PRODUCTION OF TRYPTOPHAN-DERIVED PRODUCTS TPH1, TPH2, SLC6A4 ADRA2A 400/4885ADRA2B 846/4885ADRA2C 785/4885
US-12303520-B2 Aqueous nebulization composition PDE12, CYP11B2, IL5 ADRA2A 270/4885ADRA2B 81/4885ADRA2C 31/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.